SCHEMBL8370522

SCHEMBL8370522

COc1ccc(NC2=CC(=O)c3nc(-c4ccccc4)c(-c4ccccc4)nc3C2=O)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 2/20 0.57
IDO1 P14902 2/20 0.50
MAPT P10636 7/20 0.49
LMNA P02545 2/20 0.49
MAPK1 P28482 2/20 0.49
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 3/20 0.47
NPSR1 Q6W5P4 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
PTGDR2 Q9Y5Y4 1/20 0.46
RAB9A P51151 3/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
NPC1 O15118 2/20 0.45
ALOX12 P18054 1/20 0.45
HSD17B10 Q99714 1/20 0.45
CDK1 P06493 1/20 0.45
KDR P35968 1/20 0.45
ADORA2A P29274 1/20 0.44
ADORA2B P29275 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8367237 0.87 MAPT (0.55) CDK4IDO1MAPTLMNAMAPK1
SCHEMBL8368915 0.84 CDK4 (0.65) CDK4IDO1MAPTLMNAMAPK1
SCHEMBL8368813 0.83 CDK4 (0.53) CDK4IDO1MAPTLMNAMAPK1
SCHEMBL8369508 0.78 CDK4 (0.60) CDK4IDO1MAPTLMNAMAPK1
SCHEMBL8371662 0.76 CDK4 (0.50) CDK4IDO1MAPTALDH1A1TDP1
SCHEMBL8367064 0.76 CDK4 (0.62) CDK4IDO1MAPTLMNAMAPK1
SCHEMBL16296903 0.74 MAPT (0.69) CDK4IDO1MAPTLMNAMAPK1
SCHEMBL29633276 0.74 MAPT (0.69) CDK4IDO1MAPTLMNAMAPK1
SCHEMBL10506975 0.73 ALDH1A1 (0.71) CDK4IDO1MAPTLMNAMAPK1
SCHEMBL19409875 0.73 MAPT (0.61) CDK4IDO1MAPTLMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999052365-A1 ANTICANCER AGENTS ELI LILLY AND COMPANY (US) 1999-10-21 WO disclosed