SCHEMBL8375669

SCHEMBL8375669

CCc1ccc(-c2ccc(C#N)cc2)c(-c2ccccc2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.55
KDM1A O60341 4/20 0.44
MAPT P10636 2/20 0.44
ALDH1A1 P00352 2/20 0.44
MAPK1 P28482 2/20 0.44
NPC1 O15118 1/20 0.44
LMNA P02545 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
TSHR P16473 2/20 0.43
HSD17B10 Q99714 1/20 0.43
CYP11B2 P19099 3/20 0.42
KDM4E B2RXH2 1/20 0.41
IDO1 P14902 1/20 0.41
GABRA1 P14867 1/20 0.40
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40
GABRA5 P31644 1/20 0.40
GABRA3 P34903 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8375672 0.85 PTGDR2 (0.44) CYP2A6ALDH1A1MAPK1TSHRHSD17B10
SCHEMBL8459740 0.85 MAPT (0.57) CYP2A6MAPTALDH1A1MAPK1NPC1
SCHEMBL4651878 0.84 TSHR (0.62) CYP2A6KDM1ATSHRHSD17B10CYP19A1
SCHEMBL4604750 0.84 TSHR (0.62) CYP2A6KDM1ATSHRHSD17B10CYP19A1
SCHEMBL30266947 0.84 TSHR (0.62) CYP2A6KDM1ATSHRHSD17B10CYP19A1
SCHEMBL4603532 0.83 TSHR (0.65) KDM1ATSHRHSD17B10CYP19A1
SCHEMBL9632643 0.83 TSHR (0.65) KDM1ATSHRHSD17B10CYP19A1
SCHEMBL11730491 0.83 TSHR (0.65) KDM1ATSHRHSD17B10CYP19A1
SCHEMBL4605460 0.83 TSHR (0.65) KDM1ATSHRHSD17B10CYP19A1
SCHEMBL11572123 0.83 TSHR (0.65) KDM1ATSHRHSD17B10CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5958290-A ELECTROOPTICAL APPARATUS WITH DIELECTRIC LIQUID CRYSTALS FOR RADIATION TRANSPARENT MEDIUM MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1999-09-28 US disclosed
US-5344587-A Nitriles MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1994-09-06 US disclosed