SCHEMBL8377372

SCHEMBL8377372

C=C(C)c1cc(C#N)ccc1N1CC(=O)NC1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.37
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NSD2 O96028 1/20 0.34
OPRL1 P41146 2/20 0.33
OPRM1 P35372 1/20 0.33
SLC6A9 P48067 1/20 0.33
SLC6A5 Q9Y345 1/20 0.33
BRD4 O60885 2/20 0.32
BTK Q06187 1/20 0.32
BRD2 P25440 1/20 0.32
HSD17B3 P37058 1/20 0.32
SETDB1 Q15047 1/20 0.32
LMNA P02545 1/20 0.32
GABRA1 P14867 1/20 0.32
GABRG2 P18507 1/20 0.32
GABRB3 P28472 1/20 0.32
GABRA5 P31644 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8379317 0.76 CASP3 (0.38) CASP3KDM4EALDH1A1MAPTSMN1; SMN2
SCHEMBL6740517 0.70 POLB (0.46) KDM4EMAPTOPRL1OPRM1
SCHEMBL8380654 0.70 SRD5A1 (0.38) NSD2OPRL1OPRM1
SCHEMBL3559706 0.69 NSD2 (0.58) NSD2
SCHEMBL23013861 0.69 NOS3 (0.39) KDM4EALDH1A1
SCHEMBL7394220 0.68 KDM4E (0.41) CASP3KDM4EALDH1A1MAPTSMN1; SMN2
SCHEMBL8377427 0.68 NAMPT (0.41) OPRL1OPRM1GABRA1GABRG2GABRB3
SCHEMBL7395289 0.68 KDM4E (0.39) CASP3KDM4EALDH1A1MAPTSMN1; SMN2
SCHEMBL4781539 0.68 KDM4E (0.48) CASP3KDM4EALDH1A1MAPTSMN1; SMN2
SCHEMBL7388593 0.68 IDO1 (0.34) KDM4EALDH1A1MAPTSMN1; SMN2NSD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5863947-A Phenylglycine derivatives useful for treating disorders of the central nervous system ELI LILLY AND COMPANY LIMITED (GB) 1999-01-26 US disclosed