SCHEMBL8378573

SCHEMBL8378573

Cc1ccc(S(=O)(=O)OCCc2ccccc2C2OCCO2)cc1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA9 Q16790 1/20 0.37
HTR6 P50406 1/20 0.36
VDR P11473 1/20 0.35
FFAR4 Q5NUL3 1/20 0.35
ALDH1A1 P00352 3/20 0.35
TAAR1 Q96RJ0 1/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
PSMD10 O75832 1/20 0.34
CYP24A1 Q07973 1/20 0.34
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
CYP3A4 P08684 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8518530 0.94 CA12 (0.34) CA12CA1CA9HTR6VDR
SCHEMBL9690321 0.85 CA12 (0.34) CA12CA1CA9HTR6VDR
SCHEMBL12676668 0.78 MEN1 (0.51) CA12CA1CA9VDRALDH1A1
SCHEMBL18926552 0.77 PSMD10 (0.45) CA12CA1CA9VDRALDH1A1
SCHEMBL17320652 0.76 HTR6 (0.52) HTR6VDRALDH1A1MEN1KMT2A
SCHEMBL2568984 0.76 ALDH1A1 (0.48) CA12CA1CA9VDRALDH1A1
SCHEMBL1904847 0.76 VDR (0.40) CA12CA1CA9VDRALDH1A1
SCHEMBL28774223 0.76 MEN1 (0.46) CA12CA1CA9VDRTAAR1
SCHEMBL5748460 0.76 LMNA (0.48) CA12CA1CA9VDRALDH1A1
SCHEMBL8209789 0.76 TP53 (0.51) VDRALDH1A1TAAR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5883102-A Pharmaceutically active compounds ASTRA PHARMACEUTICALS LIMITED (GB) 1999-03-16 US disclosed
EP-0858451-A1 PHARMACEUTICALLY ACTIVE QUINAZOLINE COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-08-19 EP disclosed
WO-1997014686-A1 PHARMACEUTICALLY ACTIVE QUINAZOLINE COMPOUNDS ASTRA PHARMACEUTICALS LIMITED (GB) 1997-04-24 WO disclosed