SCHEMBL8380944

SCHEMBL8380944

O=C(O)[C@H]1NC(=S)O[C@@H]1c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 2/20 0.37
TDP1 Q9NUW8 2/20 0.35
ALDH1A1 P00352 2/20 0.35
EDNRA P25101 1/20 0.35
KDM4E B2RXH2 1/20 0.35
PKM P14618 1/20 0.35
HPGD P15428 1/20 0.35
ALOX12 P18054 1/20 0.35
RAB9A P51151 1/20 0.35
HSPA1A P0DMV8 1/20 0.35
PTPN7 P35236 1/20 0.35
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
POLB P06746 1/20 0.33
CASP6 P55212 1/20 0.33
CYP2D6 P10635 1/20 0.33
CA2 P00918 1/20 0.33
HTT P42858 1/20 0.33
DHFR P00374 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8895580 0.82 CYP2D6 (0.47) TDP1ALDH1A1KMT2APOLBCYP2D6
SCHEMBL9321602 0.81 GRM5 (0.46) EPHX1TDP1ALDH1A1EDNRAKDM4E
SCHEMBL7527637 0.81 GRM5 (0.46) EPHX1TDP1ALDH1A1EDNRAKDM4E
SCHEMBL8895590 0.79 CA1 (0.39) TDP1ALDH1A1KDM4EHPGDALOX12
SCHEMBL8977701 0.72 SLC6A2 (0.46) EPHX1TDP1ALDH1A1KDM4EPKM
SCHEMBL7899177 0.69 CYP2C9 (0.43) TDP1ALDH1A1KDM4EHSPA1APTPN7
SCHEMBL11546959 0.68 CYP2D6 (0.46) EPHX1TDP1ALDH1A1KDM4EKMT2A
SCHEMBL7534121 0.68 GRM5 (0.44) EPHX1KDM4ERAB9AMAPTPOLB
SCHEMBL6509232 0.66 EDNRA (0.47) ALDH1A1EDNRAKDM4EHPGDRAB9A
SCHEMBL8345851 0.66 SLC1A2 (0.30) KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0425212-B1 Cyclic anti-aggregatory peptides SMITHKLINE BEECHAM CORP (US) 1999-04-07 EP disclosed
EP-0425212-A2 Cyclic anti-aggregatory peptides SMITHKLINE BEECHAM CORPORATION (US) 1991-05-02 EP disclosed