SCHEMBL8392000

SCHEMBL8392000

Cn1c(=O)[nH]c(N)c(NC(=O)Cc2ccccc2)c1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
GAA P10253 2/20 0.45
KDM4E B2RXH2 1/20 0.45
EPHX2 P34913 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.43
HPGD P15428 2/20 0.43
ADORA2B P29275 2/20 0.41
BRPF1 P55201 2/20 0.41
CNR2 P34972 1/20 0.41
RAB9A P51151 4/20 0.41
NPC1 O15118 3/20 0.41
KMT2A Q03164 2/20 0.40
KCNQ2 O43526 1/20 0.40
PKM P14618 1/20 0.40
MAPK1 P28482 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CYP1A2 P05177 2/20 0.40
CYP2C19 P33261 2/20 0.40
MAPT P10636 1/20 0.40
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8394013 0.84 NLRP3 (0.46) ALDH1A1EPHX2ADORA2BCNR2POLB
SCHEMBL3983281 0.79 NLRP3 (0.46) ALDH1A1GAAKDM4EEPHX2SMN1; SMN2
SCHEMBL4406872 0.79 ALDH1A1 (0.53) ALDH1A1GAAKDM4ESMN1; SMN2HPGD
SCHEMBL3447830 0.74 MAPT (0.42) ALDH1A1GAAKDM4ESMN1; SMN2ADORA2B
SCHEMBL3979338 0.72 PCK1 (0.47) GAAKDM4EKMT2AMAPTPOLB
SCHEMBL13541545 0.67 HPGD (0.70) ALDH1A1GAAEPHX2SMN1; SMN2HPGD
SCHEMBL30378242 0.66 EPHX2 (0.54) ALDH1A1EPHX2SMN1; SMN2HPGDRAB9A
SCHEMBL16028787 0.66 ALDH1A1 (0.43) ALDH1A1GAAKDM4ESMN1; SMN2HPGD
SCHEMBL17377336 0.65 EGFR (0.36) ALDH1A1GAAKDM4EHPGDADORA2B
SCHEMBL2271787 0.65 L3MBTL1 (0.47) ALDH1A1GAAKDM4ESMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5939419-A HYPOTENSIVE AGENTS AND BRONCHODILATOR AGENTS SCHERING-PLOUGH CORPORATION (US) 1999-08-17 US disclosed
EP-0686157-A1 2-BENZYL-POLYCYCLIC GUANINE DERIVATIVES AND PROCESS FOR PREPARING THEM SCHERING CORPORATION (US) 1995-12-13 EP disclosed
WO-1994019351-A1 2-BENZYL-POLYCYCLIC GUANINE DERIVATIVES AND PROCESS FOR PREPARING THEM SCHERING CORPORATION (US) 1994-09-01 WO disclosed