SCHEMBL8395016

SCHEMBL8395016

Cc1ccccc1Oc1ccc([N+](=O)[O-])cc1C(O)P(=O)(O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBXA2R P21731 4/20 0.49
HSPB1 P04792 1/20 0.41
GRIN2D O15399 1/20 0.41
GRIN3B O60391 1/20 0.41
GRIN1 Q05586 1/20 0.41
GRIN2A Q12879 1/20 0.41
GRIN2B Q13224 1/20 0.41
GRIN2C Q14957 1/20 0.41
GRIN3A Q8TCU5 1/20 0.41
CA12 O43570 2/20 0.40
CA1 P00915 2/20 0.40
MMP2 P08253 2/20 0.40
ACP3 P15309 1/20 0.40
MAPT P10636 3/20 0.39
NPSR1 Q6W5P4 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8398440 0.88 GRIN2D (0.41) TBXA2RGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL8397457 0.84 MAPT (0.46) TBXA2RHSPB1GRIN2DGRIN3BGRIN1
SCHEMBL8397454 0.82 ALDH1A1 (0.46) TBXA2RHSPB1GRIN2DGRIN3BGRIN1
SCHEMBL8394842 0.82 TBXA2R (0.48) TBXA2RHSPB1GRIN2DGRIN3BGRIN1
SCHEMBL8398648 0.81 TBXA2R (0.51) TBXA2RGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL8398452 0.81 TDP1 (0.51) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL8398658 0.79 ALDH1A1 (0.51) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL22966296 0.79 TBXA2R (0.56) TBXA2RHSPB1MAPTNPSR1CYP1A2
SCHEMBL8395390 0.77 PDE7A (0.48) TBXA2RHSPB1GRIN2DGRIN3BGRIN1
SCHEMBL8398691 0.77 TBXA2R (0.46) TBXA2RHSPB1GRIN2DGRIN3BGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5994563-A THIOPHENE DERIVATIVES, IMMUNOSUPPRESSANTS ORTHO PHARMACEUTICAL CORPORATION (US) 1999-11-30 US disclosed