SCHEMBL8395266

SCHEMBL8395266

Cc1ccc(CCNC(=O)c2ccc(NC(=N)N3CCCC3)cc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.59
NAMPT P43490 7/20 0.54
NPC1 O15118 3/20 0.54
RAB9A P51151 3/20 0.54
TP53 P04637 3/20 0.54
NPSR1 Q6W5P4 1/20 0.54
MCHR1 Q99705 5/20 0.53
CHRM1 P11229 2/20 0.53
HTR2A P28223 2/20 0.53
CYP2D6 P10635 1/20 0.53
SMN1; SMN2 Q16637 2/20 0.52
LMNA P02545 3/20 0.49
KDM4E B2RXH2 1/20 0.48
MEN1 O00255 1/20 0.48
MAPT P10636 1/20 0.48
KMT2A Q03164 1/20 0.48
MCL1 Q07820 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8525511 0.88 NAMPT (0.57) NAMPTNPC1RAB9AMCHR1CHRM1
SCHEMBL8392950 0.87 KDM1A (0.53) ALDH1A1NAMPTNPC1RAB9ATP53
Hydrochloric Acid SCHEMBL8392052 0.86 KDM1A (0.52) ALDH1A1NPC1RAB9ATP53NPSR1
SCHEMBL8524910 0.82 NAMPT (0.64) NAMPTNPC1RAB9ASMN1; SMN2
SCHEMBL8523428 0.81 NAMPT (0.60) NAMPTNPC1RAB9A
SCHEMBL3875743 0.80 MCHR1 (0.80) ALDH1A1NPC1RAB9ANPSR1MCHR1
SCHEMBL8524903 0.79 NAMPT (0.67) NAMPTTP53MCHR1CHRM1HTR2A
SCHEMBL14469162 0.78 NPC1 (0.84) ALDH1A1NAMPTNPC1RAB9ATP53
SCHEMBL11485841 0.78 RAB9A (0.62) ALDH1A1NPC1RAB9ANPSR1CYP2D6
Iodide SCHEMBL11484015 0.77 RAB9A (0.60) ALDH1A1NPC1RAB9ANPSR1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0690851-B1 GUANIDINE DERIVATIVES USEFUL IN THERAPY ASTRA AB (SE) 1999-05-19 EP claimed
US-5885985-A Guanidine derivatives useful in therapy ASTRA AKTIEBOLAG (SE) 1999-03-23 US claimed
EP-0690851-A1 GUANIDINE DERIVATIVES USEFUL IN THERAPY Astra Aktiebolag (SE) 1996-01-10 EP claimed
WO-1994021621-A1 GUANIDINE DERIVATIVES USEFUL IN THERAPY ASTRA AKTIEBOLAG (SE) 1994-09-29 WO claimed
US-5998399-A Guanidine derivatives useful in therapy as inhibitors of nitric oxide synthetase ASTRA AKTIEBOLAG (SE) 1999-12-07 US disclosed
EP-0690851-B1 GUANIDINE DERIVATIVES USEFUL IN THERAPY ASTRA AB (SE) 1999-05-19 EP disclosed
US-5885985-A Guanidine derivatives useful in therapy ASTRA AKTIEBOLAG (SE) 1999-03-23 US disclosed