SCHEMBL8525511

SCHEMBL8525511

N=C(Nc1ccc(C(=O)NCCc2ccccc2)cc1)N1CCCC1

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 8/20 0.57
HDAC2 Q92769 2/20 0.54
HDAC8 Q9BY41 1/20 0.54
HDAC6 Q9UBN7 1/20 0.54
HDAC1 Q13547 1/20 0.54
NPC1 O15118 3/20 0.53
RAB9A P51151 3/20 0.53
MCHR1 Q99705 3/20 0.52
CYP2D6 P10635 1/20 0.52
CHRM1 P11229 1/20 0.52
HTR2A P28223 1/20 0.52
GAA P10253 1/20 0.51
GALR1 P47211 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8524910 0.93 NAMPT (0.64) NAMPTNPC1RAB9A
SCHEMBL8523428 0.92 NAMPT (0.60) NAMPTNPC1RAB9A
SCHEMBL8395266 0.88 ALDH1A1 (0.59) NAMPTNPC1RAB9AMCHR1CYP2D6
SCHEMBL8396226 0.88 ALDH1A1 (0.56) NAMPTHDAC2HDAC8HDAC6RAB9A
SCHEMBL8394017 0.87 LMNA (0.58) NAMPTHDAC2HDAC8HDAC6HDAC1
Hydrochloric Acid SCHEMBL8397090 0.86 LMNA (0.57) NAMPTHDAC2HDAC8HDAC6HDAC1
SCHEMBL8524903 0.85 NAMPT (0.67) NAMPTMCHR1CYP2D6CHRM1HTR2A
SCHEMBL8394079 0.81 NPC1 (0.54) NAMPTNPC1RAB9A
SCHEMBL8392136 0.81 GAA (0.46) NAMPTNPC1RAB9AGAA
Hydrochloric Acid SCHEMBL8395526 0.80 NPC1 (0.53) NAMPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5885985-A Guanidine derivatives useful in therapy ASTRA AKTIEBOLAG (SE) 1999-03-23 US claimed
US-5885985-A Guanidine derivatives useful in therapy ASTRA AKTIEBOLAG (SE) 1999-03-23 US disclosed