SCHEMBL8395346

SCHEMBL8395346

CCCCON(C(N)=O)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.44
LMNA P02545 3/20 0.44
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
NR1I2 O75469 1/20 0.44
CHRM2 P08172 1/20 0.44
ADRA2A P08913 1/20 0.44
MAPT P10636 1/20 0.44
OPRK1 P41145 1/20 0.44
HTR2B P41595 1/20 0.44
SLC6A3 Q01959 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
TSHR P16473 5/20 0.44
TDP1 Q9NUW8 3/20 0.44
L3MBTL1 Q9Y468 3/20 0.44
ALDH1A1 P00352 4/20 0.43
MAPK1 P28482 2/20 0.43
HSD17B10 Q99714 1/20 0.42
NPC1 O15118 1/20 0.40
JAK2 O60674 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18554188 0.95 CYP3A4 (0.50) CYP3A4LMNAKMT2AMEN1NR1I2
SCHEMBL27399370 0.94 LMNA (0.52) CYP3A4LMNAKMT2AMEN1NR1I2
Formaldehyde SCHEMBL28509743 0.92 CYP3A4 (0.48) CYP3A4LMNAKMT2AMEN1NR1I2
SCHEMBL6002982 0.87 TSHR (0.46) CYP3A4LMNAKMT2ATSHRTDP1
SCHEMBL6002978 0.85 TSHR (0.45) CYP3A4LMNAKMT2ATSHRTDP1
SCHEMBL8395345 0.84 TSHR (0.44) CYP3A4LMNAKMT2ATSHRTDP1
SCHEMBL8396605 0.84 ALDH1A1 (0.43) CYP3A4LMNAKMT2AMEN1NR1I2
SCHEMBL5510643 0.83 ALDH1A1 (0.44) LMNAKMT2AMEN1MAPTTSHR
SCHEMBL6003625 0.83 L3MBTL1 (0.49) CYP3A4KMT2ACHRM2MAPTTSHR
SCHEMBL6001172 0.82 TSHR (0.47) CYP3A4LMNAKMT2AMEN1NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5864043-A CARDIOVASCULAR DISORDERS AND ANGIOTENSIN ANTAGONIST KARL THOMAE GMBH (DE) 1999-01-26 US disclosed
US-5541229-A ANGIOITENSIN II ANTAGONIST AS HYPOTENSIVE AGENTS, ANTIISCHEMIC AGENTS AND CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1996-07-30 US disclosed