SCHEMBL8398142

SCHEMBL8398142

S=c1[nH]c(=S)n(CC2CCCCC2)c2nc[nH]c12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MPO P05164 6/20 0.52
TPO P07202 4/20 0.52
CDK2 P24941 5/20 0.37
CDK1 P06493 4/20 0.37
CCNB1 P14635 3/20 0.37
CCNA2 P20248 3/20 0.37
CCNA1 P78396 3/20 0.37
CCNB2 O95067 1/20 0.37
MAPK3 P27361 1/20 0.37
CLK1 P49759 1/20 0.37
CDK5 Q00535 1/20 0.37
PIN1 Q13526 1/20 0.37
CCNB3 Q8WWL7 1/20 0.37
MAP3K5 Q99683 1/20 0.37
MTOR P42345 4/20 0.37
PIK3CA P42336 1/20 0.37
GSK3A P49840 1/20 0.37
TDP1 Q9NUW8 1/20 0.36
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8396841 0.93 MPO (0.52) MPOTPOTDP1PDE4AADORA2A
SCHEMBL1460900 0.87 MPO (0.69) MPOTPOMTORPIK3CAGSK3A
SCHEMBL1461291 0.80 MPO (0.70) MPOTPOPDE4AADORA2APDE4B
SCHEMBL10978398 0.76 PDE4A (0.59) MPOTPOMTORPIK3CAGSK3A
SCHEMBL8000339 0.75 ADORA2A (0.54) MPOTPOTDP1PDE4AADORA2A
SCHEMBL1387996 0.75 ADORA1 (0.43) ADORA2A
SCHEMBL7025705 0.74 ADORA2B (0.55) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL9350679 0.73 PDE4A (0.54) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL8002258 0.73 PDE4A (0.56) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL7021175 0.72 ADORA2B (0.56) PDE4AADORA2APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0916672-A1 6-Amino purine derivatives having PDE-IV inhibition activity and intermediates Euroceltique S.A. (LU) 1999-05-19 EP disclosed
EP-0916673-A1 6-Amino purine derivatives having PDE-IV inhibition activity Euroceltique S.A. (LU) 1999-05-19 EP disclosed