SCHEMBL8398581

SCHEMBL8398581

COc1cccc(Oc2c(Cl)nc(-c3ccco3)nc2OS(=O)(=O)c2ccc(C)cn2)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPBWR1 P48145 1/20 0.35
MCHR1 Q99705 1/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
POLB P06746 2/20 0.35
TP53 P04637 1/20 0.35
PIN1 Q13526 1/20 0.34
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
HPGD P15428 2/20 0.33
RAB9A P51151 2/20 0.33
EDNRB P24530 1/20 0.33
EDNRA P25101 1/20 0.33
DHPS P49366 1/20 0.33
NPC1 O15118 1/20 0.33
MAPT P10636 2/20 0.32
SIRT1 Q96EB6 1/20 0.32
ADORA3 P0DMS8 2/20 0.32
ADORA2A P29274 2/20 0.32
ADORA1 P30542 2/20 0.32
MEN1 O00255 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8398843 0.87 DHPS (0.41) SMN1; SMN2POLBTP53ALDH1A1EDNRB
SCHEMBL7580836 0.84 EDNRA (0.44) EDNRBEDNRA
SCHEMBL7589698 0.78 ALDH1A1 (0.47) SMN1; SMN2POLBTP53KDM4EALDH1A1
SCHEMBL8398732 0.77 EDNRA (0.42) EDNRBEDNRADHPS
SCHEMBL7591508 0.75 EDNRA (0.54) EDNRBEDNRA
SCHEMBL7589754 0.74 EDNRA (0.47) EDNRBEDNRA
SCHEMBL8399583 0.73 EDNRA (0.51) EDNRBEDNRA
SCHEMBL8399581 0.73 EDNRA (0.44) EDNRBEDNRA
SCHEMBL7585609 0.68 EDNRB (0.51) EDNRBEDNRA
SCHEMBL7582159 0.68 HPGD (0.47) SMN1; SMN2POLBTP53KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5856484-A Sulfonylaminopyrimidine carboxylic acid derivatives having endothelin inhibiting activity HOFFMANN-LA ROCHE INC. (US) 1999-01-05 US disclosed