SCHEMBL8399083

SCHEMBL8399083

Fc1ccc2nc(CNc3ccccc3Br)sc2c1F

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.34
ERBB2 P04626 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 4/20 0.33
HTT P42858 1/20 0.33
NAAA Q02083 1/20 0.32
AKR1B1 P15121 2/20 0.32
TRPM5 Q9NZQ8 1/20 0.31
RAB9A P51151 2/20 0.31
MAPT P10636 2/20 0.31
LMNA P02545 1/20 0.31
HPGD P15428 1/20 0.31
KMT2A Q03164 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
LCK P06239 1/20 0.30
SCN1A P35498 1/20 0.30
SCN5A Q14524 1/20 0.30
SCN8A Q9UQD0 1/20 0.30
NPC1 O15118 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8399168 0.89 L3MBTL1 (0.38) GSK3BERBB2KDM4EALDH1A1HTT
SCHEMBL8399102 0.86 MEN1 (0.36) GSK3BERBB2KDM4ETRPM5MAPT
SCHEMBL8398164 0.86 ADRA2C (0.40) GSK3BERBB2ALDH1A1HTTNAAA
SCHEMBL8397939 0.84 ADRA1D (0.40) GSK3BKDM4EALDH1A1NAAAAKR1B1
SCHEMBL8395190 0.83 L3MBTL1 (0.44) GSK3BERBB2ALDH1A1HTTRAB9A
SCHEMBL8399066 0.82 CYP1A2 (0.35) KDM4EALDH1A1NAAAAKR1B1RAB9A
SCHEMBL8395348 0.81 AKR1B1 (0.39) ERBB2KDM4EALDH1A1HTTAKR1B1
SCHEMBL8396103 0.81 AKR1B1 (0.41) GSK3BERBB2KDM4EALDH1A1HTT
SCHEMBL8396660 0.80 MEN1 (0.36) ERBB2ALDH1A1HTTTRPM5RAB9A
SCHEMBL8395427 0.79 EGFR (0.38) ERBB2MAPTKMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647636-B1 BENZOTHIAZOLE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF SENJU PHARMA CO (JP) 1999-06-09 EP disclosed
US-5532257-A ENZYME INHIBITOR SENJU PHARMACEUTICAL CO., LTD (JP) 1996-07-02 US disclosed
EP-0647636-A1 BENZOTHIAZOLE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF Senju Pharmaceutical Co., Ltd. (JP) 1995-04-12 EP disclosed