SCHEMBL8396103

SCHEMBL8396103

Fc1cc(F)c2sc(CNc3ccccc3Br)nc2c1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 9/20 0.41
HTT P42858 1/20 0.35
GSK3B P49841 1/20 0.33
ERBB2 P04626 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 2/20 0.32
MAPT P10636 1/20 0.32
SCN1A P35498 1/20 0.32
SCN5A Q14524 1/20 0.32
SCN8A Q9UQD0 1/20 0.32
NPC1 O15118 1/20 0.32
POLB P06746 1/20 0.32
RAB9A P51151 1/20 0.32
ABCG2 Q9UNQ0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8395524 0.90 AKR1B1 (0.43) AKR1B1HTTGSK3BKDM4EALDH1A1
SCHEMBL8396268 0.86 AKR1B1 (0.41) AKR1B1HTTALDH1A1MAPTNPC1
SCHEMBL8395800 0.86 AKR1B1 (0.41) AKR1B1
SCHEMBL8399286 0.84 AKR1B1 (0.39) AKR1B1KDM4EALDH1A1MAPTPOLB
SCHEMBL8399103 0.83 L3MBTL1 (0.43) AKR1B1HTTKDM4EALDH1A1MAPT
SCHEMBL8399351 0.83 AKR1B1 (0.46) AKR1B1MAPTNPC1RAB9A
SCHEMBL8395435 0.81 AKR1B1 (0.38) AKR1B1HTTALDH1A1MAPTNPC1
SCHEMBL8399083 0.81 GSK3B (0.34) AKR1B1HTTGSK3BERBB2KDM4E
SCHEMBL8399092 0.80 AKR1B1 (0.38) AKR1B1ERBB2
SCHEMBL8398073 0.80 AKR1B1 (0.45) AKR1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647636-B1 BENZOTHIAZOLE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF SENJU PHARMA CO (JP) 1999-06-09 EP disclosed
US-5532257-A ENZYME INHIBITOR SENJU PHARMACEUTICAL CO., LTD (JP) 1996-07-02 US disclosed
EP-0647636-A1 BENZOTHIAZOLE COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE THEREOF Senju Pharmaceutical Co., Ltd. (JP) 1995-04-12 EP disclosed