SCHEMBL839910

SCHEMBL839910

CCCCC(=O)N(CCNC(=O)[C@@H](CS)CC(C)C)Cc1ccc(-c2ccccc2S(=O)(=O)NC(=O)[C@H](C)O)c(Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 12/20 0.37
AGTR2 P50052 3/20 0.37
MME P08473 10/20 0.36
ALDH1A1 P00352 1/20 0.34
BLM P54132 1/20 0.34
LTB4R2 Q9NPC1 2/20 0.34
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
NCOR2 Q9Y618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL840591 0.96 AGTR1 (0.37) AGTR1AGTR2MME
SCHEMBL840866 0.90 AGTR1 (0.43) AGTR1AGTR2MMELTB4R2
SCHEMBL840212 0.89 AGTR1 (0.36) AGTR1AGTR2MME
SCHEMBL839142 0.88 MME (0.40) AGTR1AGTR2MMEALDH1A1BLM
SCHEMBL839141 0.88 MME (0.40) AGTR1AGTR2MMEALDH1A1BLM
SCHEMBL838701 0.86 AGTR1 (0.36) AGTR1AGTR2MME
SCHEMBL838700 0.86 AGTR1 (0.36) AGTR1AGTR2MME
SCHEMBL2975994 0.85 AGTR2 (0.40) AGTR1AGTR2ALDH1A1BLMLTB4R2
SCHEMBL839968 0.85 AGTR1 (0.38) AGTR1AGTR2MME
SCHEMBL839967 0.85 AGTR1 (0.38) AGTR1AGTR2MME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143298-B2 Dual-acting antihypertensive agents THERAVANCE, INC. (US) 2012-03-27 US disclosed