SCHEMBL8399106

SCHEMBL8399106

COC(=O)N[C@@H](C(C)C)C(O)C1C(=O)C1c1ccccc1

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33
TAS1R2 Q8TE23 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
ALDH1A1 P00352 3/20 0.33
POLB P06746 2/20 0.33
EDNRA P25101 1/20 0.33
HTRA1 Q92743 1/20 0.32
MAPT P10636 2/20 0.32
CYP2C9 P11712 1/20 0.32
TSHR P16473 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8394419 0.81 KMT2A (0.36) SMN1; SMN2TAS1R3TAS1R1TAS1R2TDP1
SCHEMBL7343203 0.79 CYP1A2 (0.48) MEN1KMT2A
Hydrochloric Acid SCHEMBL7337135 0.72 ALDH1A1 (0.36) KDM1ASMN1; SMN2ALDH1A1EDNRAMAPT
SCHEMBL8397312 0.69 CYP2D6 (0.42) MAPT
SCHEMBL8399100 0.67 ADORA3 (0.35) SMN1; SMN2TDP1ALDH1A1MAPTCYP2C9
SCHEMBL10052320 0.65 CYP2D6 (0.40) SMN1; SMN2TAS1R3TAS1R1TAS1R2ALDH1A1
SCHEMBL20055159 0.64 CYP2D6 (0.41) SMN1; SMN2TAS1R3TAS1R1TAS1R2
SCHEMBL20622277 0.64 CYP2D6 (0.41) SMN1; SMN2TAS1R3TAS1R1TAS1R2
SCHEMBL14853205 0.62 HDAC1 (0.57) ALDH1A1POLBMAPTCYP2C9TSHR
SCHEMBL31159159 0.62 NPC1 (0.53) ALDH1A1MAPTCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0590650-B1 Cyclopropene derivatives with thiol protease inhibiting activity MITSUBISHI CHEM CORP (JP) 1999-05-26 EP disclosed
US-5395958-A Intermediates for enzyme inhibitors MITSUBISHI KASEI CORPORATION (JP) 1995-03-07 US disclosed
EP-0590650-A1 Cyclopropene derivatives with thiol protease inhibiting activity Mitsubishi Chemical Corporation (JP) 1994-04-06 EP disclosed