SCHEMBL7343203

SCHEMBL7343203

CC(C)[C@H](NC(=O)[C@H](C)NC(=O)OCc1ccccc1)C(O)C1C(=O)C1c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.48
CTSK P43235 7/20 0.47
CTSL P07711 2/20 0.45
CTSS P25774 2/20 0.45
CTSB P07858 1/20 0.45
MEN1 O00255 1/20 0.44
LMNA P02545 1/20 0.44
KMT2A Q03164 1/20 0.44
ELANE P08246 2/20 0.43
PSMB8 P28062 1/20 0.42
PSMB9 P28065 1/20 0.42
PSMB5 P28074 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7339599 1.00 CYP1A2 (0.48) CYP1A2CTSKCTSLCTSSCTSB
SCHEMBL7337136 0.89 CTSL (0.52) CTSKCTSLCTSSCTSB
SCHEMBL7337274 0.82 PSMB1 (0.49) CTSKCTSLCTSSCTSBPSMB5
SCHEMBL8399106 0.79 KDM1A (0.34) MEN1KMT2A
SCHEMBL10706457 0.77 CTSK (0.55) CYP1A2CTSKCTSLCTSSCTSB
SCHEMBL11515552 0.75 CTSK (0.63) CYP1A2CTSKCTSLCTSSCTSB
SCHEMBL10612913 0.75 CTSK (0.63) CYP1A2CTSKCTSLCTSSCTSB
SCHEMBL22753446 0.75 CTSK (0.63) CYP1A2CTSKCTSLCTSSCTSB
SCHEMBL7339604 0.74 CTSK (0.50) CYP1A2CTSKCTSLCTSSCTSB
SCHEMBL7343207 0.74 CTSK (0.50) CYP1A2CTSKCTSLCTSSCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5416117-A Protease inhibitor MITSUBISHI KASEI CORPORATION (JP) 1995-05-16 US disclosed
EP-0520427-B1 Cyclopropenone derivatives MITSUBISHI CHEM IND (JP) 1994-12-14 EP disclosed
US-5328909-A Protease inhibitors MITSUBISHI KASEI CORPORATION (JP) 1994-07-12 US disclosed
EP-0520427-A1 Cyclopropenone derivatives Mitsubishi Chemical Corporation (JP) 1992-12-30 EP disclosed