SCHEMBL8399463

SCHEMBL8399463

O=C(O)Cc1oc2ccc(Cl)cc2c1-c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.52
CA2 P00918 2/20 0.52
ADORA3 P0DMS8 2/20 0.51
KDM4E B2RXH2 4/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
TNKS O95271 1/20 0.49
MAPT P10636 2/20 0.46
ALDH1A1 P00352 4/20 0.44
HPGD P15428 2/20 0.44
HSD17B10 Q99714 2/20 0.44
AKR1B1 P15121 1/20 0.44
MAP2 P11137 2/20 0.44
MCL1 Q07820 1/20 0.43
TTR P02766 1/20 0.43
GABRP O00591 1/20 0.42
GABRD O14764 1/20 0.42
GABRA1 P14867 1/20 0.42
GABRB1 P18505 1/20 0.42
GABRG2 P18507 1/20 0.42
GABRB3 P28472 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8784721 0.84 POLB (0.48) CA1CA2ADORA3KDM4ETNKS
SCHEMBL8401455 0.83 LMNA (0.47) CA1CA2ADORA3KDM4EL3MBTL1
SCHEMBL8784504 0.83 KDM4E (0.56) CA1CA2ADORA3KDM4ETNKS
SCHEMBL8403474 0.80 LMNA (0.42) ADORA3KDM4EALDH1A1HPGDHSD17B10
Hydrochloric Acid SCHEMBL11626175 0.80 CA1 (0.55) CA1CA2ADORA3KDM4EL3MBTL1
SCHEMBL8402613 0.79 SMN1; SMN2 (0.45) CA1CA2ADORA3KDM4EL3MBTL1
SCHEMBL11545978 0.78 MCL1 (0.61) KDM4EALDH1A1HPGDHSD17B10MCL1
SCHEMBL8401426 0.78 MCL1 (0.61) CA1CA2ADORA3KDM4ETNKS
SCHEMBL28837168 0.78 CA1 (0.49) CA1CA2ADORA3KDM4EL3MBTL1
SCHEMBL25824715 0.77 ADORA3 (0.65) CA1CA2ADORA3KDM4ETNKS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5929107-A INHIBITORS OF ACYL-COA:CHOLESTEROL ACYLTRANSFERASE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-07-27 US disclosed
US-5492929-A ENZYME INHIBITORS, ANTICHOLESTEROL AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-02-20 US disclosed
EP-0602598-A1 3-Phenylindolyl-, -benzofuranyl- and -benzothienyl- alkylcarboxanilides, their production and use Takeda Chemical Industries, Ltd. (JP) 1994-06-22 EP disclosed