SCHEMBL8399570

SCHEMBL8399570

CC(=O)N(CCNC(=O)OC(C)(C)C)c1cccc(F)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.46
MAPK3 P27361 3/20 0.41
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41
MTNR1A P48039 5/20 0.41
MTNR1B P49286 5/20 0.41
NQO2 P16083 1/20 0.41
CKS1B P61024 1/20 0.40
SKP1 P63208 1/20 0.40
SKP2 Q13309 1/20 0.40
KDM4E B2RXH2 1/20 0.40
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
PTBP1 P26599 1/20 0.40
HTT P42858 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HDAC1 Q13547 1/20 0.39
HDAC8 Q9BY41 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5037820 0.80 KMT2A (0.44) CTSSCTSKNQO2ALDH1A1LMNA
SCHEMBL15584401 0.76 NQO2 (0.43) MTNR1AMTNR1BNQO2CKS1BSKP1
SCHEMBL16499930 0.76 CKS1B (0.42) MTNR1AMTNR1BNQO2CKS1BSKP1
SCHEMBL28824481 0.76 MAPK3 (0.49) MAPK3MTNR1AMTNR1BCKS1BSKP1
SCHEMBL15283620 0.76 CKS1B (0.50) CTSSMTNR1AMTNR1BNQO2CKS1B
SCHEMBL5729170 0.75 CTSS (0.54) CTSSCTSKNQO2KDM4ELMNA
SCHEMBL7578637 0.73 MTNR1A (0.46) MTNR1AMTNR1BNQO2CKS1BSKP1
SCHEMBL15584389 0.73 MAPT (0.47) MTNR1AMTNR1BNQO2CKS1BSKP1
SCHEMBL16444538 0.73 SMN1; SMN2 (0.47) CKS1BSKP1SKP2KDM4ENPC1
SCHEMBL16444539 0.73 SMN1; SMN2 (0.47) CKS1BSKP1SKP2KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5998415-A Bicyclic heteroaryl-alkylene-(homo)piperazinones and thione analogues thereof, their preparation, and their use of as selective agonists of 5-HT1 -like receptors MERCK SHARP & DOHME LTD. (GB) 1999-12-07 US disclosed