SCHEMBL839993

SCHEMBL839993

CC(C)CC(CS)C(=O)NCCN(Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1)C(=O)CC1CCCC1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.37
AGTR1 P30556 10/20 0.36
MME P08473 9/20 0.36
HTR5A P47898 5/20 0.35
HTR1A P08908 1/20 0.35
DRD2 P14416 1/20 0.35
DRD4 P21917 1/20 0.35
HTR1D P28221 1/20 0.35
HTR1B P28222 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR7 P34969 1/20 0.35
ADRA1B P35368 1/20 0.35
DRD3 P35462 1/20 0.35
HTR2B P41595 1/20 0.35
HTR6 P50406 1/20 0.35
SLC2A1 P11166 1/20 0.34
LTB4R2 Q9NPC1 1/20 0.34
MMP3 P08254 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL839257 0.97 AGTR1 (0.37) SLC6A4AGTR1MMEHTR5AHTR1A
SCHEMBL841570 0.94 SLC6A4 (0.42) SLC6A4AGTR1MMEHTR5AHTR1A
SCHEMBL839718 0.90 BACE1 (0.35) AGTR1MMEMMP3
SCHEMBL839269 0.89 AGTR1 (0.40) AGTR1MMELTB4R2
SCHEMBL840167 0.88 MLNR (0.39) AGTR1MME
SCHEMBL839172 0.88 AGTR1 (0.37) AGTR1MME
SCHEMBL839949 0.88 AGTR1 (0.41) AGTR1MMELTB4R2
SCHEMBL839252 0.88 AGTR1 (0.41) AGTR1MMELTB4R2
SCHEMBL859394 0.88 AGTR1 (0.41) AGTR1MMELTB4R2
SCHEMBL841053 0.87 REN (0.42) AGTR1MMELTB4R2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143298-B2 Dual-acting antihypertensive agents THERAVANCE, INC. (US) 2012-03-27 US disclosed