SCHEMBL8400437

SCHEMBL8400437

COc1ccc(-c2nsnc2C(=O)O)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALPL P05186 1/20 0.50
CA9 Q16790 1/20 0.50
PRKAG1 P54619 1/20 0.49
PRKAA1 Q13131 1/20 0.49
PRKAB1 Q9Y478 1/20 0.49
ALDH1A1 P00352 3/20 0.48
MAPT P10636 3/20 0.48
HPGD P15428 1/20 0.48
RECQL P46063 1/20 0.48
PTGS2 P35354 2/20 0.47
KDM4E B2RXH2 1/20 0.47
LMNA P02545 1/20 0.47
GAA P10253 1/20 0.47
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
PTGDR2 Q9Y5Y4 3/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
ATM Q13315 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8396813 0.81 ALPL (0.46) ALPLALDH1A1MAPTHPGDKDM4E
SCHEMBL8400102 0.78 CA12 (0.46) ALPLALDH1A1MAPTHPGDKDM4E
SCHEMBL8519653 0.78 CA12 (0.46) ALPLALDH1A1HPGDKDM4ELMNA
SCHEMBL30704314 0.76 ALDH1A1 (0.49) ALDH1A1MAPTHPGDPTGS2KDM4E
SCHEMBL2405190 0.75 KDM4E (0.53) ALPLCA9PRKAG1PRKAA1PRKAB1
SCHEMBL899644 0.75 BACE1 (0.52) ALDH1A1MAPTHPGDRECQLPTGS2
SCHEMBL30529887 0.74 ALDH1A1 (0.51) ALPLCA9PRKAG1PRKAA1PRKAB1
SCHEMBL8401146 0.74 MAPK1 (0.45) PTGDR2
SCHEMBL10982371 0.74 ALDH1A1 (0.50) CA9ALDH1A1MAPTHPGDRECQL
SCHEMBL10984490 0.73 ALDH1A1 (0.46) CA9ALDH1A1MAPTHPGDRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5948916-A Arylthiadiazole derivative and antiviral agent containing the same RATIONAL DRUG DESIGN LABORATORIES (JP) 1999-09-07 US disclosed
EP-0785193-A1 ARYLTHIADIAZOLE DERIVATIVE AND ANTIVIRAL AGENT CONTAINING THE SAME Rational Drug Design Laboratories (JP) 1997-07-23 EP disclosed