SCHEMBL8401146

SCHEMBL8401146

O=C(O)c1nsnc1-c1ccc(C(F)(F)F)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.45
MAP2K4 P45985 2/20 0.45
MAPK6 Q16659 2/20 0.45
MAPKAPK3 Q16644 1/20 0.45
SRD5A2 P31213 1/20 0.42
PLAU P00749 1/20 0.42
MAPKAPK5 Q8IW41 1/20 0.42
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
DHODH Q02127 3/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.40
KIF11 P52732 4/20 0.40
CYP2C8 P10632 1/20 0.40
PTGER1 P34995 1/20 0.39
RXRA P19793 1/20 0.39
RXRB P28702 1/20 0.39
RXRG P48443 1/20 0.39
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39
IKBKB O14920 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8400098 0.82 PIN1 (0.52) SRD5A2
SCHEMBL8400102 0.81 CA12 (0.46) MAPK1MAP2K4MAPK6PTGDR2
SCHEMBL10338995 0.79 KDM4E (0.52) MAPK1DHODH
SCHEMBL8519653 0.78 CA12 (0.46) MAP2K4DHODHPTGDR2
SCHEMBL8396813 0.78 ALPL (0.46) MAPK1MAP2K4MAPK6MAPKAPK3SRD5A2
SCHEMBL8400437 0.74 ALPL (0.50) PTGDR2
SCHEMBL11405709 0.73 MAPK1 (0.44) MAPK1MAP2K4MAPK6MAPKAPK3SRD5A2
SCHEMBL24987817 0.71 DHODH (0.47) MAPK1MAP2K4MAPK6MAPKAPK3SRD5A2
SCHEMBL8842879 0.71 MKNK1 (0.48) MAPK1MAP2K4MAPK6MAPKAPK3SRD5A2
SCHEMBL2467798 0.70 PLAU (0.50) MAPK1MAP2K4MAPK6MAPKAPK3SRD5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5948916-A Arylthiadiazole derivative and antiviral agent containing the same RATIONAL DRUG DESIGN LABORATORIES (JP) 1999-09-07 US disclosed
EP-0785193-A1 ARYLTHIADIAZOLE DERIVATIVE AND ANTIVIRAL AGENT CONTAINING THE SAME Rational Drug Design Laboratories (JP) 1997-07-23 EP disclosed