SCHEMBL8405232

SCHEMBL8405232

CCn1c(=O)[nH]c2c[nH]c(=O)nc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 6/20 0.46
PDE4A P27815 5/20 0.46
PDE4B Q07343 5/20 0.46
PDE4C Q08493 5/20 0.46
PDE4D Q08499 5/20 0.46
CYP1A2 P05177 3/20 0.45
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
BLM P54132 2/20 0.41
LMNA P02545 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
TSHR P16473 1/20 0.41
NFKB1 P19838 1/20 0.41
PMP22 Q01453 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ADORA2B P29275 3/20 0.35
ADORA3 P0DMS8 3/20 0.35
HPGD P15428 1/20 0.35
ADORA1 P30542 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8404996 0.84 PDE4A (0.51) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL8407924 0.78 HPGD (0.54) MEN1KMT2ALMNACYP3A4TSHR
SCHEMBL8407814 0.77 GAA (0.47) ADORA2AMEN1KMT2ALMNACYP3A4
SCHEMBL8407994 0.76 ADORA3 (0.47) MEN1KMT2ALMNATSHRSMN1; SMN2
SCHEMBL21285531 0.73 CYP1A2 (0.49) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL8407844 0.73 POLB (0.44) ADORA2BPGRPOLB
SCHEMBL8405032 0.73 KMT2A (0.46) MEN1KMT2ATSHRNFKB1POLB
SCHEMBL28642857 0.72 CYP1A2 (0.47) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL24765254 0.71 ADORA2A (0.48) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL8407979 0.71 POLB (0.33) CYP1A2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0673938-B1 Purine derivatives and pharmaceutically acceptable salts thereof NIPPON ZOKI PHARMACEUTICAL CO (JP) 1999-07-07 EP disclosed
US-5658918-A INHIBITING NASAL MUCOUS SECRETION NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 1997-08-19 US disclosed
EP-0673938-A2 Novel purine derivatives and pharmaceutically acceptable salts thereof NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 1995-09-27 EP disclosed