SCHEMBL8404996

SCHEMBL8404996

CCCCn1c(=O)[nH]c2c[nH]c(=O)nc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 4/20 0.51
ADORA2A P29274 4/20 0.51
PDE4B Q07343 4/20 0.51
PDE4C Q08493 4/20 0.51
PDE4D Q08499 4/20 0.51
ALDH1A1 P00352 6/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
BRD4 O60885 1/20 0.46
BRD2 P25440 1/20 0.46
BRD3 Q15059 1/20 0.46
BRDT Q58F21 1/20 0.46
ADORA2B P29275 3/20 0.45
ADORA3 P0DMS8 2/20 0.45
HPGD P15428 4/20 0.43
HSD17B10 Q99714 3/20 0.43
KDM4A O75164 1/20 0.43
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
CASP1 P29466 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8405232 0.84 ADORA2A (0.46) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL8407994 0.77 ADORA3 (0.47) ALDH1A1MEN1KMT2AADORA2BADORA3
SCHEMBL8407814 0.76 GAA (0.47) ADORA2AMEN1KMT2AADORA2BADORA3
SCHEMBL8407924 0.73 HPGD (0.54) ALDH1A1MEN1KMT2ABRD4ADORA3
SCHEMBL11234998 0.70 ALDH1A1 (0.52) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL4191402 0.70 PDE4A (0.45) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL8407844 0.69 POLB (0.44) ADORA2B
SCHEMBL8405032 0.69 KMT2A (0.46) ALDH1A1MEN1KMT2ATSHRCASP1
SCHEMBL7602847 0.68 PDE4A (1.00) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL14560539 0.67 ALDH1A1 (0.73) ADORA2AALDH1A1ADORA2BADORA3HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0673938-B1 Purine derivatives and pharmaceutically acceptable salts thereof NIPPON ZOKI PHARMACEUTICAL CO (JP) 1999-07-07 EP disclosed
US-5658918-A INHIBITING NASAL MUCOUS SECRETION NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 1997-08-19 US disclosed
EP-0673938-A2 Novel purine derivatives and pharmaceutically acceptable salts thereof NIPPON ZOKI PHARMACEUTICAL CO., LTD. (JP) 1995-09-27 EP disclosed