SCHEMBL8406485

SCHEMBL8406485

CCN(c1nc(F)ccc1[N+](=O)[O-])C1CCN(Cc2ccccc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.46
NPSR1 Q6W5P4 1/20 0.44
CHRM2 P08172 1/20 0.43
CHRM3 P20309 1/20 0.43
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
SIGMAR1 Q99720 2/20 0.42
MAPT P10636 1/20 0.42
PKM P14618 1/20 0.42
RAB9A P51151 1/20 0.42
OPRM1 P35372 3/20 0.42
SCN1A P35498 1/20 0.42
SCN8A Q9UQD0 1/20 0.42
ACHE P22303 2/20 0.41
FAAH O00519 1/20 0.41
BCHE P06276 1/20 0.41
BACE1 P56817 1/20 0.41
CCR4 P51679 1/20 0.41
BLM P54132 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8406779 0.88 SCN1A (0.49) MAPK1NPSR1CHRM2CHRM3KMT2A
SCHEMBL8409570 0.84 MAPK1 (0.50) MAPK1NPSR1CHRM2CHRM3KMT2A
SCHEMBL8791981 0.82 MAPK1 (0.45) MAPK1NPSR1CHRM2CHRM3KMT2A
SCHEMBL8406857 0.82 OPRM1 (0.43) SIGMAR1OPRM1SCN1ASCN8AACHE
SCHEMBL8791942 0.81 ACHE (0.50) MAPK1NPSR1CHRM2CHRM3KMT2A
SCHEMBL8410128 0.78 GMNN (0.41) SIGMAR1OPRM1SCN1ASCN8AACHE
SCHEMBL8410140 0.78 SCN1A (0.41) SIGMAR1OPRM1SCN1ASCN8AACHE
SCHEMBL8409472 0.77 MAPK1 (0.49) MAPK1NPSR1CHRM2CHRM3KMT2A
SCHEMBL8406812 0.76 CHRM2 (0.43) MAPK1CHRM2CHRM3SIGMAR1OPRM1
SCHEMBL8791696 0.76 MAPK1 (0.48) MAPK1NPSR1CHRM2CHRM3KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5866589-A Alkyl substituted piperadinyl and piperazinyl anti-AIDS compounds PHARMACIA & UPJOHN COMPANY (US) 1999-02-02 US disclosed
WO-1996018628-A1 ALKYL SUBSTITUTED PIPERADINYL AND PIPERAZINYL ANTI-AIDS COMPOUNDS PHARMACIA & UPJOHN COMPANY (US) 1996-06-20 WO disclosed