SCHEMBL8407134

SCHEMBL8407134

CCCCN(C(=O)C(C)C)c1ccc(C#N)c(C#N)c1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 9/20 0.52
ALDH1A1 P00352 2/20 0.40
HPGD P15428 1/20 0.40
PGR P06401 3/20 0.38
AR P10275 1/20 0.37
ADRB2 P07550 1/20 0.36
NOS2 P35228 1/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8407140 0.86 MLYCD (0.48) MLYCDALDH1A1HPGDPGRAR
SCHEMBL8409270 0.76 MLYCD (0.44) MLYCDALDH1A1PGRARMAOA
SCHEMBL28308819 0.75 SLC16A3 (0.42) ALDH1A1HPGDPGRARNOS2
SCHEMBL18997806 0.74 MLYCD (0.62) MLYCDALDH1A1HPGDADRB2TSHR
SCHEMBL11453144 0.70 MLYCD (0.53) MLYCDALDH1A1ADRB2
SCHEMBL3048940 0.69 AR (0.44) PGRARNOS2MAOAMAOB
SCHEMBL6843869 0.68 MLYCD (1.00) MLYCD
SCHEMBL4896904 0.68 MAOA (0.38) PGRARNOS2MAOAMAOB
SCHEMBL4896895 0.68 MAOA (0.38) PGRARNOS2MAOAMAOB
SCHEMBL4219142 0.68 PGR (0.40) MLYCDALDH1A1PGRARMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5994362-A ADMINISTERING FINASTERIDE AND CASODEX MERCK & CO., INC. (US) 1999-11-30 US disclosed
EP-0514056-A2 Use of estrogens or antiandrogens for reversal of male sexual phenotype in poultry MERCK & CO. INC. (US) 1992-11-19 EP disclosed
WO-1992016233-A1 PHARMACEUTICAL COMBINATION FOR THE TREATMENT OF PROSTATIC CANCER CONTAINING A 5 ALPHA REDUCTASE INHIBITOR AND AN ANTIANDROGEN MERCK & CO., INC. (US) 1992-10-01 WO disclosed
EP-0002309-B1 ACYLANILIDES, PROCESS FOR THEIR MANUFACTURE AND PHARMACEUTICAL AND VETERINARY COMPOSITIONS CONTAINING THEM IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1982-12-01 EP disclosed
US-4282218-A ANTIANDROGENS IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1981-08-04 US disclosed
US-4239776-A Anti-androgenic amides IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1980-12-16 US disclosed
EP-0002309-A2 Acylanilides, process for their manufacture and pharmaceutical and veterinary compositions containing them IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1979-06-13 EP disclosed