SCHEMBL8409270

SCHEMBL8409270

CC(C)C(=O)N(C)c1ccc(C#N)c(C#N)c1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 3/20 0.44
PGR P06401 3/20 0.43
AR P10275 1/20 0.41
USP30 Q70CQ3 2/20 0.40
ITK Q08881 1/20 0.38
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
CHRNB2 P17787 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNA4 P43681 1/20 0.35
XDH P47989 2/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
KCNH2 Q12809 1/20 0.33
IDE P14735 1/20 0.33
RORC P51449 1/20 0.33
SLC22A12 Q96S37 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4219142 0.88 PGR (0.40) MLYCDPGRARUSP30ITK
SCHEMBL31026325 0.83 AR (0.62) MLYCDPGRAR
SCHEMBL8407140 0.80 MLYCD (0.48) MLYCDPGRARMAOAMAOB
SCHEMBL1380362 0.78 AR (0.46) MLYCDPGRARCYP2C9
SCHEMBL8407134 0.76 MLYCD (0.52) MLYCDPGRARMAOAMAOB
SCHEMBL4901224 0.74 MAOA (0.41) PGRARMAOAMAOBALDH1A1
SCHEMBL18935755 0.72 MLYCD (0.50) MLYCDUSP30ALDH1A1
SCHEMBL15378494 0.71 MLYCD (0.47) MLYCDALDH1A1
SCHEMBL4893929 0.70 MAOA (0.41) PGRARMAOAMAOBALDH1A1
SCHEMBL28746540 0.70 MLYCD (0.46) MLYCDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0002309-B1 ACYLANILIDES, PROCESS FOR THEIR MANUFACTURE AND PHARMACEUTICAL AND VETERINARY COMPOSITIONS CONTAINING THEM IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1982-12-01 EP claimed
US-5994362-A ADMINISTERING FINASTERIDE AND CASODEX MERCK & CO., INC. (US) 1999-11-30 US disclosed
EP-0514056-A2 Use of estrogens or antiandrogens for reversal of male sexual phenotype in poultry MERCK & CO. INC. (US) 1992-11-19 EP disclosed
WO-1992016233-A1 PHARMACEUTICAL COMBINATION FOR THE TREATMENT OF PROSTATIC CANCER CONTAINING A 5 ALPHA REDUCTASE INHIBITOR AND AN ANTIANDROGEN MERCK & CO., INC. (US) 1992-10-01 WO disclosed
EP-0002309-B1 ACYLANILIDES, PROCESS FOR THEIR MANUFACTURE AND PHARMACEUTICAL AND VETERINARY COMPOSITIONS CONTAINING THEM IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1982-12-01 EP disclosed
US-4282218-A ANTIANDROGENS IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1981-08-04 US disclosed
US-4239776-A Anti-androgenic amides IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1980-12-16 US disclosed
EP-0002309-A2 Acylanilides, process for their manufacture and pharmaceutical and veterinary compositions containing them IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1979-06-13 EP disclosed