SCHEMBL8407191

SCHEMBL8407191

Oc1cc(Cl)c(OCCCCCc2ccccc2)c(Cl)c1

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 2/20 0.46
CBS P35520 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.44
IGF1R P08069 1/20 0.44
ALOX15 P16050 1/20 0.44
CNR2 P34972 2/20 0.43
CNR1 P21554 1/20 0.43
FFAR1 O14842 1/20 0.43
TDP1 Q9NUW8 1/20 0.42
PLA2G4B P0C869 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8408802 1.00 GPR84 (0.46) GPR84CBSL3MBTL1IGF1RALOX15
SCHEMBL8405941 0.98 IGF1R (0.45) GPR84CBSL3MBTL1IGF1RALOX15
SCHEMBL8408825 0.94 IDO1 (0.46) GPR84CBSL3MBTL1IGF1RALOX15
SCHEMBL8405441 0.89 HTR1A (0.42) L3MBTL1FFAR1
SCHEMBL8408594 0.88 MRGPRX4 (0.47) GPR84L3MBTL1IGF1RALOX15CNR2
SCHEMBL8405532 0.86 IGF1R (0.51) IGF1RALOX15
SCHEMBL8409415 0.83 SLC5A1 (0.40) L3MBTL1IGF1RALOX15CNR2CNR1
SCHEMBL11239759 0.83 HPGD (0.44) GPR84L3MBTL1
SCHEMBL8408121 0.83 THRA (0.49) GPR84CBSIGF1RALOX15CNR2
SCHEMBL8407967 0.82 TAAR1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5872137-A AROMATIC OXY DIHALOPRENE COMPOUNDS INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1999-02-16 US disclosed
EP-0722430-B1 DIHALOPROPENE COMPOUNDS, INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL CO (JP) 1998-10-21 EP disclosed
EP-0722430-A1 DIHALOPROPENE COMPOUNDS, INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1996-07-24 EP disclosed
WO-1996004228-A1 DIHALOPROPENE COMPOUNDS, INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1996-02-15 WO disclosed