SCHEMBL8408982

SCHEMBL8408982

COc1ccc(-c2nc3cc(OC)ccc3c(=O)n2-c2ccc(OCCCl)cc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.61
RAB9A P51151 1/20 0.58
NPSR1 Q6W5P4 1/20 0.58
HRH3 Q9Y5N1 7/20 0.56
KCNH2 Q12809 6/20 0.56
ESR1 P03372 1/20 0.51
PDE10A Q9Y233 3/20 0.49
G6PD P11413 1/20 0.49
EGFR P00533 2/20 0.48
ADRA1A P35348 1/20 0.48
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
POLB P06746 1/20 0.45
RXFP1 Q9HBX9 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8409027 0.86 ESR1 (0.72) ALDH1A1RAB9ANPSR1HRH3KCNH2
SCHEMBL8408698 0.81 HRH3 (0.57) ALDH1A1RAB9ANPSR1HRH3KCNH2
SCHEMBL8408615 0.81 HRH3 (0.57) ALDH1A1RAB9ANPSR1HRH3KCNH2
SCHEMBL31277481 0.74 ALDH1A1 (0.95) ALDH1A1RAB9ANPSR1HRH3KCNH2
SCHEMBL11104386 0.73 ADRB1 (0.62) HRH3KCNH2ADRA1APOLBRXFP1
SCHEMBL4485049 0.72 HRH3 (1.00) HRH3KCNH2ADRA1A
SCHEMBL1663473 0.72 LMNA (0.63) ALDH1A1RAB9ANPSR1HRH3KCNH2
SCHEMBL11099494 0.72 ADRB1 (0.61) HRH3KCNH2ADRA1APOLBRXFP1
SCHEMBL8411748 0.72 ALDH1A1 (0.47) ALDH1A1RAB9ANPSR1HRH3KCNH2
SCHEMBL8408638 0.72 ALDH1A1 (0.47) ALDH1A1RAB9ANPSR1HRH3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5948775-A OSTEOPOROSIS; ANTICANCER AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1999-09-07 US disclosed