SCHEMBL8409257

SCHEMBL8409257

CN(c1nc(F)ccc1NC(C)(C)C)C1CCN(Cc2ccccc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN1A P35498 13/20 0.47
SCN8A Q9UQD0 13/20 0.47
GMNN O75496 2/20 0.47
ALDH1A1 P00352 2/20 0.47
LMNA P02545 2/20 0.47
DRD2 P14416 2/20 0.47
HPGD P15428 2/20 0.47
DRD4 P21917 2/20 0.47
DRD3 P35462 2/20 0.47
PMP22 Q01453 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
TDP1 Q9NUW8 2/20 0.47
TP53 P04637 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
KDM1A O60341 1/20 0.42
RCOR1 Q9UKL0 1/20 0.42
KCNH2 Q12809 1/20 0.41
SLC2A1 P11166 1/20 0.41
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8408627 0.89 SCN1A (0.44) SCN1ASCN8AGMNNALDH1A1LMNA
SCHEMBL8410140 0.88 SCN1A (0.41) SCN1ASCN8AKDM4EGAA
SCHEMBL8409218 0.83 DRD2 (0.61) SCN1ASCN8AGMNNALDH1A1LMNA
SCHEMBL8406887 0.81 DRD2 (0.51) SCN1ASCN8AGMNNALDH1A1LMNA
SCHEMBL8409680 0.78 ACHE (0.40) SCN1ASCN8AKDM4EGAA
SCHEMBL8409401 0.77 SLC6A12 (0.42) SCN1ASCN8AGMNNALDH1A1LMNA
SCHEMBL8406779 0.77 SCN1A (0.49) SCN1ASCN8AGMNNALDH1A1LMNA
SCHEMBL8409470 0.74 DRD2 (0.53) SCN1ASCN8AGMNNALDH1A1LMNA
SCHEMBL8410128 0.73 GMNN (0.41) SCN1ASCN8AGMNNALDH1A1LMNA
SCHEMBL8406488 0.73 DRD2 (0.49) GMNNALDH1A1LMNADRD2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5866589-A Alkyl substituted piperadinyl and piperazinyl anti-AIDS compounds PHARMACIA & UPJOHN COMPANY (US) 1999-02-02 US disclosed
EP-0797576-A1 ALKYL SUBSTITUTED PIPERADINYL AND PIPERAZINYL ANTI-AIDS COMPOUNDS PHARMACIA & UPJOHN COMPANY (US) 1997-10-01 EP disclosed
WO-1996018628-A1 ALKYL SUBSTITUTED PIPERADINYL AND PIPERAZINYL ANTI-AIDS COMPOUNDS PHARMACIA & UPJOHN COMPANY (US) 1996-06-20 WO disclosed