SCHEMBL8409596

SCHEMBL8409596

O=C(O)c1[c]c2cc([N+](=O)[O-])ccc2[nH]1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
MEN1 O00255 1/20 0.50
POLB P06746 1/20 0.50
PKM P14618 1/20 0.50
NPY1R P25929 1/20 0.50
NPY2R P49146 1/20 0.50
KMT2A Q03164 1/20 0.50
MAPT P10636 3/20 0.46
GRIA1 P42261 1/20 0.45
GRIA2 P42262 1/20 0.45
GRIA3 P42263 1/20 0.45
GRIA4 P48058 1/20 0.45
TDP1 Q9NUW8 2/20 0.43
CYP3A4 P08684 1/20 0.43
ALOX15 P16050 1/20 0.43
KDM4E B2RXH2 1/20 0.42
GAA P10253 1/20 0.42
TP53 P04637 1/20 0.41
CYP19A1 P11511 1/20 0.41
CA12 O43570 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27868663 0.83 TUBB4A (0.43) ALDH1A1MEN1POLBPKMNPY1R
SCHEMBL8409653 0.80 CACNA1C (0.47) ALDH1A1MEN1POLBPKMNPY1R
SCHEMBL2072913 0.76 GRIA1 (0.49) ALDH1A1MEN1POLBPKMNPY1R
SCHEMBL10492182 0.74 GRIA1 (0.46) ALDH1A1MEN1POLBPKMNPY1R
SCHEMBL8697240 0.70 TSHR (0.42) ALDH1A1MEN1POLBPKMNPY1R
SCHEMBL1260652 0.69 HRH4 (0.60) ALDH1A1MEN1POLBPKMNPY1R
SCHEMBL1156515 0.69 HRH4 (0.60) ALDH1A1MEN1POLBPKMNPY1R
SCHEMBL8794605 0.68 HRH4 (0.59) ALDH1A1MEN1POLBPKMNPY1R
SCHEMBL6847834 0.67 ALDH1A1 (1.00) ALDH1A1MEN1POLBPKMNPY1R
SCHEMBL3035932 0.67 ALDH1A1 (0.52) ALDH1A1MEN1POLBPKMNPY1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5866589-A Alkyl substituted piperadinyl and piperazinyl anti-AIDS compounds PHARMACIA & UPJOHN COMPANY (US) 1999-02-02 US disclosed
EP-0797576-A1 ALKYL SUBSTITUTED PIPERADINYL AND PIPERAZINYL ANTI-AIDS COMPOUNDS PHARMACIA & UPJOHN COMPANY (US) 1997-10-01 EP disclosed
WO-1996018628-A1 ALKYL SUBSTITUTED PIPERADINYL AND PIPERAZINYL ANTI-AIDS COMPOUNDS PHARMACIA & UPJOHN COMPANY (US) 1996-06-20 WO disclosed