SCHEMBL8409653

SCHEMBL8409653

CCOC(=O)c1[c]c2cc([N+](=O)[O-])ccc2[nH]1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1C Q13936 5/20 0.47
CACNA1F O60840 4/20 0.47
CACNA1D Q01668 4/20 0.47
CACNA1S Q13698 4/20 0.47
ADORA3 P0DMS8 2/20 0.47
AR P10275 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
HIF1A Q16665 3/20 0.44
MAPT P10636 3/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
CYP1A2 P05177 2/20 0.44
CYP3A4 P08684 2/20 0.44
CYP2C9 P11712 2/20 0.44
CYP2C19 P33261 2/20 0.44
POLB P06746 2/20 0.44
LMNA P02545 1/20 0.44
MAPK1 P28482 1/20 0.44
GPR55 Q9Y2T6 1/20 0.44
CYP2D6 P10635 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27868663 0.86 TUBB4A (0.43) CACNA1CADORA3SMN1; SMN2HIF1AMAPT
SCHEMBL8409596 0.80 ALDH1A1 (0.50) MAPTMEN1KMT2ACYP3A4POLB
SCHEMBL6016022 0.76 TSHR (0.47) SMN1; SMN2MAPTMEN1KMT2APOLB
SCHEMBL2072913 0.75 GRIA1 (0.49) MAPTMEN1KMT2ACYP3A4POLB
SCHEMBL656156 0.74 KDM4E (0.67) CACNA1CCACNA1FCACNA1DCACNA1SADORA3
SCHEMBL16733406 0.73 ALDH1A1 (0.71) ARSMN1; SMN2MAPTMEN1KMT2A
SCHEMBL2449511 0.72 SMN1; SMN2 (0.50) CACNA1CCACNA1FCACNA1DCACNA1SADORA3
SCHEMBL394554 0.72 ALOX15 (0.64) CACNA1CCACNA1FCACNA1DCACNA1SADORA3
SCHEMBL6001705 0.72 ALDH1A1 (0.57) ARSMN1; SMN2MAPTMEN1KMT2A
SCHEMBL4948906 0.72 ALDH1A1 (0.57) ARSMN1; SMN2MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5866589-A Alkyl substituted piperadinyl and piperazinyl anti-AIDS compounds PHARMACIA & UPJOHN COMPANY (US) 1999-02-02 US disclosed
EP-0797576-A1 ALKYL SUBSTITUTED PIPERADINYL AND PIPERAZINYL ANTI-AIDS COMPOUNDS PHARMACIA & UPJOHN COMPANY (US) 1997-10-01 EP disclosed
WO-1996018628-A1 ALKYL SUBSTITUTED PIPERADINYL AND PIPERAZINYL ANTI-AIDS COMPOUNDS PHARMACIA & UPJOHN COMPANY (US) 1996-06-20 WO disclosed