SCHEMBL8409979

SCHEMBL8409979

CC(C)Nc1cc(F)ccc1N(C)C1CCN(Cc2ccccc2)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GMNN O75496 2/20 0.50
ALDH1A1 P00352 2/20 0.50
LMNA P02545 2/20 0.50
DRD2 P14416 2/20 0.50
HPGD P15428 2/20 0.50
DRD4 P21917 2/20 0.50
DRD3 P35462 2/20 0.50
PMP22 Q01453 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
TDP1 Q9NUW8 2/20 0.50
TP53 P04637 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CCR3 P51677 1/20 0.45
ACHE P22303 3/20 0.45
BACE1 P56817 3/20 0.45
BCHE P06276 2/20 0.45
SCN1A P35498 5/20 0.45
SCN8A Q9UQD0 5/20 0.45
MEN1 O00255 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9092750 0.81 ACHE (0.43) CCR3ACHEBACE1BCHESCN1A
SCHEMBL8792841 0.77 ACHE (0.49) ALDH1A1DRD2SMN1; SMN2CCR3ACHE
SCHEMBL8409470 0.75 DRD2 (0.53) GMNNALDH1A1LMNADRD2HPGD
SCHEMBL8793282 0.73 ACHE (0.47) ALDH1A1SMN1; SMN2CCR3ACHEBACE1
SCHEMBL21375648 0.71 SIGMAR1 (0.60) GMNNALDH1A1LMNADRD2HPGD
SCHEMBL7286179 0.70 ACHE (0.53) GMNNALDH1A1LMNADRD2HPGD
SCHEMBL8410128 0.70 GMNN (0.41) GMNNALDH1A1LMNADRD2HPGD
SCHEMBL2108897 0.69 ACHE (0.66) DRD2DRD4DRD3CCR3ACHE
SCHEMBL9093241 0.68 MEN1 (0.45) ALDH1A1CCR3ACHEBACE1BCHE
SCHEMBL3311545 0.68 ACHE (0.60) GMNNALDH1A1LMNADRD2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5866589-A Alkyl substituted piperadinyl and piperazinyl anti-AIDS compounds PHARMACIA & UPJOHN COMPANY (US) 1999-02-02 US disclosed
EP-0797576-A1 ALKYL SUBSTITUTED PIPERADINYL AND PIPERAZINYL ANTI-AIDS COMPOUNDS PHARMACIA & UPJOHN COMPANY (US) 1997-10-01 EP disclosed
WO-1996018628-A1 ALKYL SUBSTITUTED PIPERADINYL AND PIPERAZINYL ANTI-AIDS COMPOUNDS PHARMACIA & UPJOHN COMPANY (US) 1996-06-20 WO disclosed