SCHEMBL8410489

SCHEMBL8410489

COC(=O)CCNC(=O)c1cccc(-c2ccccc2)c1OC

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 1/20 0.56
KDM5B Q9UGL1 1/20 0.48
HPGD P15428 1/20 0.48
MAPK1 P28482 1/20 0.48
PDCD1 Q15116 1/20 0.47
CD274 Q9NZQ7 1/20 0.47
HTT P42858 2/20 0.46
CHRNB2 P17787 1/20 0.45
CHRNB4 P30926 1/20 0.45
CHRNA3 P32297 1/20 0.45
CHRNA4 P43681 1/20 0.45
TAS1R3 Q7RTX0 1/20 0.45
TAS1R1 Q7RTX1 1/20 0.45
PPARG P37231 1/20 0.44
ALDH1A1 P00352 1/20 0.44
PRSS1 P07477 1/20 0.43
CTSG P08311 1/20 0.43
CTRB1 P17538 1/20 0.43
CMA1 P23946 1/20 0.43
GAA P10253 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8410787 0.83 NR1H4 (0.62) NR1H4KDM5BHPGDMAPK1PDCD1
SCHEMBL14121014 0.77 MAPK1 (0.54) HPGDMAPK1HTTPPARGPRSS1
SCHEMBL449968 0.77 HDAC3 (0.51) NR1H4HPGDMAPK1PDCD1CD274
SCHEMBL27375291 0.76 CHRNB2 (0.54) MAPK1PDCD1CD274HTTCHRNB2
SCHEMBL4831306 0.76 NR1H4 (0.56) NR1H4HPGDPDCD1CD274HTT
SCHEMBL27890118 0.76 NR1H4 (0.56) NR1H4HTTALDH1A1GAAKDM4E
SCHEMBL30394743 0.76 HNF4A (0.58) NR1H4HPGDMAPK1HTTALDH1A1
SCHEMBL4632581 0.76 HNF4A (0.58) NR1H4HPGDMAPK1HTTALDH1A1
SCHEMBL2662273 0.75 CNR1 (0.42) HPGDHTT
SCHEMBL17799595 0.74 HNF4A (0.56) NR1H4HPGDMAPK1HTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5922763-A ANTICOAGULANT; CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1999-07-13 US disclosed