SCHEMBL8410787

SCHEMBL8410787

COc1c(C(=O)NCC(=O)O)cccc1-c1ccccc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 1/20 0.62
KEAP1 Q14145 1/20 0.53
KDM4E B2RXH2 2/20 0.49
HPGD P15428 2/20 0.49
ALDH1A1 P00352 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
HTT P42858 1/20 0.49
CHRNB2 P17787 2/20 0.48
CHRNA4 P43681 2/20 0.48
CHRNB4 P30926 1/20 0.48
CHRNA3 P32297 1/20 0.48
TP53 P04637 1/20 0.47
TAS1R3 Q7RTX0 1/20 0.47
TAS1R1 Q7RTX1 1/20 0.47
GAA P10253 2/20 0.46
POLB P06746 1/20 0.46
KDM6B O15054 1/20 0.45
FTO Q9C0B1 1/20 0.45
EGLN1 Q9GZT9 1/20 0.45
KDM4C Q9H3R0 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8410489 0.83 NR1H4 (0.56) NR1H4KDM4EHPGDALDH1A1HTT
SCHEMBL10788983 0.82 HPGD (0.49) KEAP1KDM4EHPGDALDH1A1SMN1; SMN2
SCHEMBL1649572 0.82 CHRNB2 (0.68) KEAP1ALDH1A1HTTCHRNB2CHRNA4
SCHEMBL436284 0.81 KEAP1 (0.57) KEAP1ALDH1A1HTTCHRNB2CHRNA4
SCHEMBL4831306 0.79 NR1H4 (0.56) NR1H4KDM4EHPGDALDH1A1SMN1; SMN2
SCHEMBL30394743 0.79 HNF4A (0.58) NR1H4KDM4EHPGDALDH1A1SMN1; SMN2
SCHEMBL4632581 0.79 HNF4A (0.58) NR1H4KDM4EHPGDALDH1A1SMN1; SMN2
SCHEMBL27890118 0.79 NR1H4 (0.56) NR1H4KDM4EALDH1A1SMN1; SMN2HTT
SCHEMBL17799595 0.77 HNF4A (0.56) NR1H4KDM4EHPGDALDH1A1SMN1; SMN2
SCHEMBL27450922 0.77 KEAP1 (0.66) KEAP1KDM4EALDH1A1HTTCHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5922763-A ANTICOAGULANT; CARDIOVASCULAR DISORDERS DR. KARL THOMAE GMBH (DE) 1999-07-13 US disclosed
US-5736559-A CARDIOVASCULAR DISORDERS; RESPIRATORY SYSTEM DISORDERS KARL THOMAE GMBH (DE) 1998-04-07 US disclosed