SCHEMBL8412919

SCHEMBL8412919

COc1cc(C)cc(Sc2cccc(F)c2C#N)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 6/20 0.36
IDO1 P14902 2/20 0.36
ACHE P22303 1/20 0.36
MAPT P10636 2/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
PGR P06401 1/20 0.35
ALDH1A1 P00352 2/20 0.35
HTR1A P08908 1/20 0.34
HTR3A P46098 1/20 0.34
DRD2 P14416 1/20 0.34
HTR2A P28223 1/20 0.34
HRH1 P35367 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
SQOR Q9Y6N5 1/20 0.34
KDM4E B2RXH2 1/20 0.34
HPGD P15428 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8410372 0.89 AR (0.40) ARIDO1MAPTLMNAHTT
SCHEMBL8410613 0.86 DHFR (0.44) ARIDO1MAPTLMNAHTT
SCHEMBL8643800 0.86 ALDH1A1 (0.39) ARIDO1ACHEMAPTHTT
SCHEMBL9014990 0.83 AR (0.36) ARMAPTLMNASMN1; SMN2PGR
SCHEMBL1154616 0.82 L3MBTL1 (0.44) ARIDO1ACHEMAPTLMNA
SCHEMBL2075358 0.79 L3MBTL1 (0.42) ARMAPTLMNAPGRALDH1A1
SCHEMBL8647963 0.77 ADORA2A (0.42) ARIDO1MAPTHTTALDH1A1
SCHEMBL8569510 0.76 DHFR (0.44) ARIDO1ACHEMAPTSMN1; SMN2
SCHEMBL8642759 0.72 CYP19A1 (0.42) IDO1MAPTLMNAHTTSMN1; SMN2
SCHEMBL8644586 0.72 KDM4E (0.45) ARIDO1MAPTHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0748311-B1 THERAPEUTIC BENZONITRILES WELLCOME FOUND (GB) 1999-08-04 EP disclosed
US-5723452-A Therapeutic benzonitriles GLAXO WELLCOME INC. (US) 1998-03-03 US disclosed
EP-0748311-A1 THERAPEUTIC BENZONITRILES THE WELLCOME FOUNDATION LIMITED (GB) 1996-12-18 EP disclosed
WO-1995023133-A1 THERAPEUTIC BENZONITRILES THE WELLCOME FOUNDATION LIMITED (GB) 1995-08-31 WO disclosed