SCHEMBL8410372

SCHEMBL8410372

Cc1cc(C)cc(Sc2cccc(F)c2C#N)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 4/20 0.40
PGR P06401 1/20 0.40
KDM4E B2RXH2 5/20 0.37
ALDH1A1 P00352 5/20 0.37
HPGD P15428 2/20 0.37
HSD17B10 Q99714 1/20 0.37
L3MBTL1 Q9Y468 3/20 0.34
TDP1 Q9NUW8 2/20 0.34
MAPT P10636 2/20 0.34
LMNA P02545 2/20 0.34
PKM P14618 1/20 0.34
POLB P06746 2/20 0.33
HTR1A P08908 2/20 0.33
HTR3A P46098 2/20 0.33
KMT2A Q03164 2/20 0.33
DRD2 P14416 1/20 0.33
HTR2A P28223 1/20 0.33
HRH1 P35367 1/20 0.33
TUBB4A P04350 1/20 0.33
TUBB P07437 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9014990 0.90 AR (0.36) ARPGRKDM4EALDH1A1HPGD
SCHEMBL1154616 0.89 L3MBTL1 (0.44) ARPGRKDM4EALDH1A1HPGD
SCHEMBL8412919 0.89 AR (0.36) ARPGRKDM4EALDH1A1HPGD
SCHEMBL2075358 0.86 L3MBTL1 (0.42) ARPGRKDM4EALDH1A1HPGD
SCHEMBL8644586 0.81 KDM4E (0.45) ARKDM4EALDH1A1HPGDL3MBTL1
SCHEMBL9015004 0.77 AR (0.42) ARPGRKDM4EALDH1A1HPGD
SCHEMBL8410613 0.77 DHFR (0.44) ARPGRKDM4EALDH1A1HPGD
SCHEMBL1154522 0.76 MAOA (0.47) ARPGRKDM4EALDH1A1HPGD
SCHEMBL8641570 0.76 TDP1 (0.40) KDM4EALDH1A1HSD17B10TDP1MAPT
SCHEMBL846222 0.74 ALDH1A1 (0.41) ARPGRKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0748311-B1 THERAPEUTIC BENZONITRILES WELLCOME FOUND (GB) 1999-08-04 EP disclosed
US-5723452-A Therapeutic benzonitriles GLAXO WELLCOME INC. (US) 1998-03-03 US disclosed
EP-0748311-A1 THERAPEUTIC BENZONITRILES THE WELLCOME FOUNDATION LIMITED (GB) 1996-12-18 EP disclosed
WO-1995023133-A1 THERAPEUTIC BENZONITRILES THE WELLCOME FOUNDATION LIMITED (GB) 1995-08-31 WO disclosed