Isosorbide

Isosorbide

SCHEMBL8414428

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nearest known ligand 0.56

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Isosorbide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.56
LMNA P02545 1/20 0.56
MAPT P10636 1/20 0.56
ALDH1A1 P00352 1/20 0.38
BCHE P06276 4/20 0.33
GSR P00390 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Isosorbide SCHEMBL27944142 0.89 THRB (0.65) THRBLMNAMAPTALDH1A1BCHE
Isosorbide SCHEMBL3388024 0.84 THRB (0.65) THRBLMNAMAPTALDH1A1BCHE
Isosorbide SCHEMBL4353400 0.84 THRB (0.65) THRBLMNAMAPTALDH1A1BCHE
Isosorbide SCHEMBL2129898 0.84 THRB (0.65) THRBLMNAMAPTALDH1A1BCHE
Isosorbide Mononitrate SCHEMBL8414427 0.82 MAPT (0.87) THRBLMNAMAPTALDH1A1BCHE
Isosorbide SCHEMBL24465084 0.75 THRB (1.00) THRBLMNAMAPTBCHE
Isosorbide SCHEMBL5884995 0.75 THRB (1.00) THRBLMNAMAPTBCHE
Isosorbide SCHEMBL2599531 0.75 THRB (1.00) THRBLMNAMAPTBCHE
Isosorbide SCHEMBL12504733 0.75 THRB (1.00) THRBLMNAMAPTBCHE
Isosorbide SCHEMBL15495 0.75 THRB (1.00) THRBLMNAMAPTBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0936901-A1 PHARMACEUTICAL COMPOSITION FOR RAPID SUSPENSION IN AQUEOUS MEDIA EURAND INTERNATIONAL S.P.A. (IT) 1999-08-25 EP claimed
WO-1998017250-A1 PHARMACEUTICAL COMPOSITION FOR RAPID SUSPENSION IN AQUEOUS MEDIA EURAND INTERNATIONAL S.P.A. (IT) 1998-04-30 WO claimed
EP-0936901-A1 PHARMACEUTICAL COMPOSITION FOR RAPID SUSPENSION IN AQUEOUS MEDIA EURAND INTERNATIONAL S.P.A. (IT) 1999-08-25 EP disclosed
WO-1998017250-A1 PHARMACEUTICAL COMPOSITION FOR RAPID SUSPENSION IN AQUEOUS MEDIA EURAND INTERNATIONAL S.P.A. (IT) 1998-04-30 WO disclosed