Isosorbide

Isosorbide

SCHEMBL27944142

O=[N+]([O-])[O-].O[C@@H]1CO[C@H]2[C@@H]1OC[C@@H]2O.[Na+]

nearest known ligand 0.65

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Isosorbide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
THRB known ✓ P10828 1/20 0.65
CA2 known ✓ P00918 1/20 0.32
LMNA P02545 1/20 0.65
MAPT P10636 1/20 0.62
ALDH1A1 P00352 1/20 0.41
GSR P00390 3/20 0.33
BCHE P06276 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Isosorbide SCHEMBL2129898 0.90 THRB (0.65) THRBLMNAMAPTALDH1A1GSR
Isosorbide SCHEMBL3388024 0.90 THRB (0.65) THRBLMNAMAPTALDH1A1GSR
Isosorbide SCHEMBL4353400 0.90 THRB (0.65) THRBLMNAMAPTALDH1A1GSR
Isosorbide SCHEMBL5699287 0.90 THRB (0.65) THRBLMNAMAPTALDH1A1GSR
Isosorbide SCHEMBL5170125 0.90 THRB (0.65) THRBLMNAMAPTALDH1A1GSR
Isosorbide SCHEMBL217707 0.90 THRB (0.65) THRBLMNAMAPTALDH1A1GSR
Isosorbide SCHEMBL8414428 0.89 THRB (0.56) THRBLMNAMAPTALDH1A1GSR
Isosorbide SCHEMBL24465084 0.81 THRB (1.00) THRBLMNAMAPTBCHE
Isosorbide SCHEMBL9882796 0.81 THRB (1.00) THRBLMNAMAPTBCHE
Isosorbide SCHEMBL6105354 0.81 THRB (1.00) THRBLMNAMAPTBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110407846-B Preparation method of 5-isosorbide mononitrate 鲁南制药集团股份有限公司 2021-09-14 CN disclosed
CN-103641840-A Method for synthesizing and purifying 5-isosorbide mononitrate QINGDAO HUANGHAI PHARMACEUTICAL CO LTD 2014-03-19 CN disclosed