SCHEMBL8416210

SCHEMBL8416210

NC(N)=NC(=O)c1ccccc1Cl

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.54
CES2 O00748 1/20 0.54
CES1 P23141 1/20 0.54
SLC9A1 P19634 4/20 0.53
ALDH1A1 P00352 2/20 0.52
HTR2B P41595 3/20 0.49
ADRA2A P08913 2/20 0.49
MEN1 O00255 1/20 0.49
LMNA P02545 1/20 0.49
CYP3A4 P08684 1/20 0.49
HTR1A P08908 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
ADRA2B P18089 1/20 0.49
ADRA2C P18825 1/20 0.49
MAOA P21397 1/20 0.49
ADRA1D P25100 1/20 0.49
HTR2A P28223 1/20 0.49
HTR2C P28335 1/20 0.49
MAPK1 P28482 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8390599 0.98 KDM4E (0.57) KDM4ECES2CES1SLC9A1ALDH1A1
Hydrochloric Acid SCHEMBL8391039 0.83 TSHR (0.53) KDM4ESLC9A1ALDH1A1HTR2BADRA2A
SCHEMBL8668407 0.78 HTR2B (0.55) SLC9A1ALDH1A1HTR2BADRA2AMEN1
SCHEMBL13017375 0.77 CES2 (0.60) KDM4ECES2CES1ALDH1A1MEN1
SCHEMBL263770 0.76 CES2 (0.65) KDM4ECES2CES1ALDH1A1MEN1
SCHEMBL29843413 0.76 CES2 (0.65) KDM4ECES2CES1ALDH1A1MEN1
Hydrochloric Acid SCHEMBL7942184 0.76 ADRA2A (0.56) KDM4ESLC9A1ALDH1A1HTR2BADRA2A
SCHEMBL14607348 0.76 SLC9A1 (0.51) SLC9A1HTR2BHTR7NPC1RAB9A
Hydrochloric Acid SCHEMBL8392499 0.76 SLC9A1 (0.56) SLC9A1ALDH1A1HTR2BHTR7RAB9A
Hydrochloric Acid SCHEMBL8393886 0.76 SMN1; SMN2 (0.53) KDM4ESLC9A1ALDH1A1HTR2BLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1064954-C Orthosubstituted benzoylguanidine, preparation of same, pharmaceutical containing same and application of same HOECHST AG (DE) 2001-04-25 CN claimed
EP-0640588-B1 Orthosubstituted benzoylguanidines, process for their preparation, their use as a medicament or diagnostic agent and a medicament containing them HOECHST AG (DE) 1999-09-08 EP claimed