SCHEMBL8417601

SCHEMBL8417601

CN1C(=O)c2ccc[n+]([O-])c2Cc2ncccc21

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TTR P02766 1/20 0.36
CES1 P23141 1/20 0.36
BRD4 O60885 12/20 0.35
ALDH1A1 P00352 2/20 0.35
HTT P42858 1/20 0.35
HSD17B10 Q99714 1/20 0.35
ADORA3 P0DMS8 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
NPC1 O15118 1/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
CA1 P00915 2/20 0.32
CA2 P00918 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8420764 0.82 TTR (0.43) TTRCES1BRD4ALDH1A1HTT
SCHEMBL12060497 0.72 BRPF1 (0.43) BRD4ALDH1A1HTTADORA3ADORA2A
SCHEMBL14099507 0.71 ADORA3 (0.37) ADORA3ADORA2AADORA1SMN1; SMN2CA1
SCHEMBL8337979 0.69 ALDH1A1 (0.39) TTRCES1BRD4ALDH1A1ADORA3
SCHEMBL8337573 0.68 ADORA3 (0.34) TTRCES1BRD4ALDH1A1HTT
SCHEMBL8790761 0.66 TTR (0.50) TTRCES1BRD4ALDH1A1HTT
SCHEMBL24440815 0.66 ADORA3 (0.33) ADORA3ADORA2AADORA1
SCHEMBL8304689 0.65 ALDH1A1 (0.52) TTRCES1BRD4ALDH1A1HTT
SCHEMBL18635357 0.64 CYP11B2 (0.44) ADORA3ADORA2AADORA1
SCHEMBL27027255 0.64 HTR2C (0.42) SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5908841-A 5,11-dihydro-6H-dipyrido 3,2-b:2',3'-e!azepine-6-ones and their use in the prevention of treatment of HIV infection BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 1999-06-01 US disclosed