SCHEMBL8419441

SCHEMBL8419441

COc1ccc(NS(=O)(=O)c2ccccc2)c(-c2ccc(OC)c(F)c2)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.48
ABCC1 P33527 1/20 0.48
KIT P10721 1/20 0.47
LMNA P02545 3/20 0.46
ACLY P53396 6/20 0.45
STAT3 P40763 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
HPGD P15428 2/20 0.45
KDM4E B2RXH2 2/20 0.45
ALDH1A1 P00352 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
AXL P30530 1/20 0.45
TSHR P16473 1/20 0.45
AAK1 Q2M2I8 1/20 0.45
PTGS1 P23219 2/20 0.44
PTGS2 P35354 2/20 0.44
MAP2K4 P45985 1/20 0.44
KEAP1 Q14145 1/20 0.44
NFE2L2 Q16236 1/20 0.44
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8421023 0.88 LMNA (0.48) ABCB1ABCC1KITLMNAACLY
SCHEMBL8421215 0.87 ACLY (0.49) LMNAACLYSMN1; SMN2HPGDKDM4E
SCHEMBL8421017 0.87 TSHR (0.46) ABCB1ABCC1KITLMNASTAT3
SCHEMBL8421287 0.80 ACLY (0.50) ABCB1ABCC1LMNAACLYSTAT3
SCHEMBL8659801 0.79 STAT3 (0.69) LMNAACLYSTAT3HPGDL3MBTL1
SCHEMBL8659675 0.78 STAT3 (0.58) ABCB1ABCC1LMNAACLYSTAT3
SCHEMBL8421183 0.76 LMNA (0.48) LMNAACLYSMN1; SMN2KDM4EALDH1A1
SCHEMBL6169842 0.76 PTGS2 (0.47) KITALDH1A1TSHRPTGS1PTGS2
SCHEMBL8478641 0.76 PTGS2 (0.44) ABCB1ABCC1KITACLYSTAT3
SCHEMBL8478256 0.74 PTGS2 (0.42) ABCB1ABCC1KITAAK1PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5916905-A ANTIARTHRITIC AGENTS; ANALGESICS; ANTIPYRETICS G. D. SEARLE & CO. (US) 1999-06-29 US disclosed
US-5686470-A 2, 3-substituted pyridines for the treatment of inflammation WEIER RICHARD M (US) 1997-11-11 US disclosed