SCHEMBL8419832

SCHEMBL8419832

O=C(OCC(Cl)(Cl)Cl)c1ccccc1C#CC1C(O)C2CCN1CC2

nearest known ligand 0.31

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.31
GABRG2 P18507 1/20 0.31
GABRB3 P28472 1/20 0.31
GABRA5 P31644 1/20 0.31
GABRA3 P34903 1/20 0.31
GABRA2 P47869 1/20 0.31
GABRA4 P48169 1/20 0.31
GABRA6 Q16445 1/20 0.31
MRGPRX1 Q96LB2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8417764 0.86 HPGD (0.34)
SCHEMBL8419750 0.85 SMN1; SMN2 (0.34) MRGPRX1
SCHEMBL8969934 0.70 MMP13 (0.46)
SCHEMBL8520797 0.70 FFAR1 (0.38)
SCHEMBL27408212 0.68 TSHR (0.55) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL8919982 0.66 MMP13 (0.46)
SCHEMBL8420487 0.65 TSHR (0.31)
SCHEMBL8419827 0.65 CYP2D6 (0.31) MRGPRX1
SCHEMBL8919905 0.63 FDFT1 (0.41)
SCHEMBL8442126 0.63 TDP1 (0.61)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5919793-A QUINUCLIDINE DERIVATIVES, SQUALENE SYNTHETASE INHIBITORS, ANTICHOLESTEROL AGENTS ZENECA LIMITED (GB) 1999-07-06 US disclosed