SCHEMBL8420280

SCHEMBL8420280

COCCOc1ccc(C#CC2C(O)C3CCN2CC3)c(CO)c1

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.33
USP30 Q70CQ3 1/20 0.32
FFAR4 Q5NUL3 1/20 0.32
CHEK2 O96017 1/20 0.31
HTR1A P08908 2/20 0.31
CYP2D6 P10635 2/20 0.31
SLC6A4 P31645 2/20 0.31
OPRM1 P35372 1/20 0.30
LRRK2 Q5S007 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8417915 0.82 ACACB (0.37) HRH3USP30CYP2D6OPRM1
SCHEMBL8417740 0.75 HRH3 (0.34) HRH3FFAR4CHEK2HTR1ACYP2D6
SCHEMBL8421884 0.74 KDM4E (0.34) SLC6A4
SCHEMBL8419842 0.73 HTR1A (0.34) HTR1A
SCHEMBL8420485 0.73 FDFT1 (0.36)
SCHEMBL8921318 0.72 ALDH1A1 (0.45) HRH3CYP2D6
SCHEMBL8422069 0.72 CTSK (0.42) HTR1A
SCHEMBL8421763 0.72 EGFR (0.34) HRH3
SCHEMBL8969567 0.71 FDFT1 (0.51)
Hydrochloric Acid SCHEMBL8919722 0.71 ALDH1A1 (0.44) HRH3CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5919793-A QUINUCLIDINE DERIVATIVES, SQUALENE SYNTHETASE INHIBITORS, ANTICHOLESTEROL AGENTS ZENECA LIMITED (GB) 1999-07-06 US disclosed