SCHEMBL8420712

SCHEMBL8420712

CCC(C)(C)Nc1c(C(N)c2cc3cc(C#N)ccc3o2)c(=O)c1=O

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 1/20 0.39
ABCC8 Q09428 1/20 0.39
KCNJ11 Q14654 1/20 0.39
KCNJ8 Q15842 1/20 0.39
PGR P06401 3/20 0.32
HRH3 Q9Y5N1 2/20 0.31
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31
DRD2 P14416 1/20 0.31
DRD4 P21917 1/20 0.31
DRD3 P35462 1/20 0.31
CYP2A6 P11509 1/20 0.31
CETP P11597 4/20 0.31
PLAU P00749 1/20 0.30
GPR35 Q9HC97 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8421284 0.87 CCR2 (0.34) ABCC9ABCC8KCNJ11KCNJ8PGR
SCHEMBL8420167 0.82 ABCC9 (0.48) ABCC9ABCC8KCNJ11KCNJ8PGR
SCHEMBL8386573 0.79 HRH3 (0.39) ABCC9ABCC8KCNJ11KCNJ8PGR
SCHEMBL4261010 0.78 ABCC9 (0.40) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8624266 0.69 AR (0.33) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL20559738 0.69 CYP2A6 (0.46) PGRHRH3NOS3NOS1NOS2
SCHEMBL8895911 0.69 CYP2A6 (0.46) PGRHRH3NOS3NOS1NOS2
SCHEMBL8665101 0.69 ABCC9 (0.37) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL8381744 0.68 HRH3 (0.40) ABCC9ABCC8KCNJ11KCNJ8PGR
SCHEMBL8622441 0.68 PDK1 (0.38) ABCC9ABCC8KCNJ11KCNJ8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5872139-A MUSCLE RELAXANTS USED TO TREAT URINARY INCONTINENCE, IRRITABLE BOWEL SYNDROME, ASTHMA, PREMATURE LABOR, CONGESTIVE HEART FAILURE, ANGINA, CEREBRAL VASCULAR DISEASE AND HYPERTENSION AMERICAN HOME PRODUCTS CORPORATION (US) 1999-02-16 US claimed
US-5872139-A MUSCLE RELAXANTS USED TO TREAT URINARY INCONTINENCE, IRRITABLE BOWEL SYNDROME, ASTHMA, PREMATURE LABOR, CONGESTIVE HEART FAILURE, ANGINA, CEREBRAL VASCULAR DISEASE AND HYPERTENSION AMERICAN HOME PRODUCTS CORPORATION (US) 1999-02-16 US disclosed