SCHEMBL8422007

SCHEMBL8422007

C=CCc1cc(CC(=O)O)ccc1O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 5/20 0.58
POLB P06746 4/20 0.58
MAPT P10636 4/20 0.58
HPGD P15428 3/20 0.58
TDP1 Q9NUW8 3/20 0.58
TSHR P16473 2/20 0.58
NFKB1 P19838 2/20 0.58
KDM4E B2RXH2 2/20 0.58
LMNA P02545 2/20 0.58
RGS12 O14924 1/20 0.58
APEX1 P27695 1/20 0.58
THPO P40225 1/20 0.58
BLM P54132 1/20 0.58
GNAI1 P63096 1/20 0.58
PMP22 Q01453 1/20 0.58
HIF1A Q16665 1/20 0.58
HSD17B10 Q99714 1/20 0.58
GABRA1 P14867 4/20 0.56
GABRB2 P47870 4/20 0.56
CA2 P00918 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10388117 0.85 GAA (0.59) GAAPOLBMAPTHPGDTDP1
SCHEMBL8418481 0.84 GABRA1 (0.53) GAAPOLBMAPTHPGDKDM4E
SCHEMBL18694877 0.83 ALDH1A1 (0.53) GAAPOLBMAPTHPGDKDM4E
SCHEMBL821126 0.82 GABRA1 (0.72) GAAPOLBMAPTHPGDKDM4E
SCHEMBL10825727 0.82 GAA (0.70) GAAPOLBMAPTHPGDTDP1
SCHEMBL7041553 0.81 ALDH1A1 (0.57) GAAPOLBMAPTHPGDKDM4E
SCHEMBL6180947 0.81 GABRA1 (0.61) GAAPOLBMAPTHPGDKDM4E
SCHEMBL16245950 0.81 GABRA1 (0.61) GAAPOLBMAPTHPGDKDM4E
SCHEMBL11278615 0.81 PTGDR (0.42) GAAPOLBMAPTHPGDTDP1
SCHEMBL10388295 0.81 GAA (0.54) GAAPOLBMAPTHPGDTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5919793-A QUINUCLIDINE DERIVATIVES, SQUALENE SYNTHETASE INHIBITORS, ANTICHOLESTEROL AGENTS ZENECA LIMITED (GB) 1999-07-06 US disclosed
EP-0696284-A1 HETEROCYCLIC DERIVATIVES ZENECA LIMITED (GB) 1996-02-14 EP disclosed
WO-1994025459-A1 HETEROCYCLIC DERIVATIVES ZENECA LIMITED (GB) 1994-11-10 WO disclosed
US-4918092-A Leukotriene antagonists MERCK FROSST CANADA, INC. (CA) 1990-04-17 US disclosed