SCHEMBL8423635

SCHEMBL8423635

O=S(=O)(Nn1nc(-c2ccc(Cl)cc2)cc1-c1ccccn1)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.43
LMNA P02545 2/20 0.42
KDM4E B2RXH2 2/20 0.42
KDM1A O60341 3/20 0.42
KAT6A Q92794 3/20 0.42
PTGS2 P35354 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
NPC1 O15118 1/20 0.41
MAPT P10636 1/20 0.41
RAB9A P51151 1/20 0.41
HTR6 P50406 1/20 0.41
PTGS1 P23219 1/20 0.40
GAA P10253 1/20 0.39
HTT P42858 1/20 0.39
DCTPP1 Q9H773 1/20 0.38
OXTR P30559 1/20 0.38
AVPR1A P37288 1/20 0.38
MAOA P21397 1/20 0.38
APP P05067 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8420848 0.91 PTGS2 (0.46) AURKALMNAKDM4EKDM1AKAT6A
SCHEMBL8421776 0.88 KDM1A (0.47) AURKAKDM4EKDM1AKAT6APTGS2
SCHEMBL8641119 0.87 AURKA (0.46) AURKAKDM4EKDM1AKAT6APTGS2
SCHEMBL8421619 0.85 KMO (0.46) AURKAKDM1APTGS2NPC1MAPT
SCHEMBL8422269 0.85 PGR (0.44) AURKALMNAKDM1AKAT6APTGS2
SCHEMBL8420906 0.85 KDM1A (0.46) AURKAKDM1APTGS2NPC1MAPT
SCHEMBL8422366 0.85 KDM1A (0.46) AURKAKDM1APTGS2NPC1MAPT
SCHEMBL8421656 0.84 KDM1A (0.42) AURKAKDM4EKDM1AKAT6APTGS2
SCHEMBL8422316 0.84 KDM1A (0.44) AURKAKDM4EKDM1APTGS2NPC1
SCHEMBL8424131 0.83 KDM1A (0.41) AURKAKDM1APTGS2MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5908852-A 1,3,5 trisubstituted pyrazole compounds for treatment of inflammation G. D. SEARLE & CO. (US) 1999-06-01 US disclosed