SCHEMBL8423709

SCHEMBL8423709

Cc1ccc(S(=O)(=O)O)cc1.N=C(Nc1ccccc1)c1ccccc1

nearest known ligand 0.51

Known targets — ChEMBL curated mechanism

ABL1BMXBRAFBTKCHRNA4CHRNB2CSNK1EEGFRERBB2F10FLT1FLT3FLT4IGF1RINSRITKJAK3KDRKITOPRM1PARP1PARP2PDGFRBPIK3CDRAF1RETSLC18A2TECTXKdacAdacBdacCftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.51
CYP2D6 P10635 2/20 0.50
MAPK1 P28482 1/20 0.50
ALDH1A1 P00352 6/20 0.48
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
NFKB1 P19838 1/20 0.48
CASP3 P42574 1/20 0.48
NFKB2 Q00653 1/20 0.48
RELA Q04206 1/20 0.48
SENP8 Q96LD8 1/20 0.48
SENP7 Q9BQF6 1/20 0.48
SENP6 Q9GZR1 1/20 0.48
HPGD P15428 3/20 0.48
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA9 Q16790 1/20 0.47
MAPT P10636 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4853047 0.82 NPC1 (0.61) LMNAALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL2154879 0.82 NPC1 (0.52) LMNAALDH1A1NPC1RAB9ASMN1; SMN2
Diphenylamine SCHEMBL3206649 0.79 GAA (0.65) LMNACYP2D6MAPK1ALDH1A1SMN1; SMN2
SCHEMBL5593961 0.78 MGLL (0.57) HPGDCA12CA1CA2CA9
SCHEMBL5595197 0.77 PTGS2 (0.54) LMNAALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL4854992 0.77 PTGS2 (0.54) LMNAALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL13836876 0.77 SMN1; SMN2 (0.73) LMNACYP2D6MAPK1ALDH1A1SMN1; SMN2
SCHEMBL932442 0.77 SMN1; SMN2 (0.73) LMNACYP2D6MAPK1ALDH1A1SMN1; SMN2
Toluene SCHEMBL180606 0.77 SMN1; SMN2 (0.65) LMNACYP2D6MAPK1ALDH1A1SMN1; SMN2
Hno SCHEMBL3391939 0.77 GAA (0.56) LMNACYP2D6MAPK1ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5237045-A Heat-resistant polytriazines using acid salts of aromatic amines as catalysts for aromatic tetracyano monomers; kinetics THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE NAVY (US) 1993-08-17 US claimed
US-20190284341-A1 3-OXO-2-ALKYLISOINDOLINE DIPHTHALONITRILE MONOMERS, METHODS OF MANUFACTURE, THERMOSETTING COMPOSITIONS COMPRISING THE SAME, AND USES THEREOF SHPP GLOBAL TECHNOLOGIES B.V. (NL) 2019-09-19 US disclosed
US-20190284339-A1 THERMOSET 3-OXO-ISOINDOLINE DIPHTHALONITRILE POLYMERS, METHOD OF MANUFACTURE, AND USES THEREOF SHPP GLOBAL TECHNOLOGIES B.V. (NL) 2019-09-19 US disclosed
US-20190284340-A1 3-OXO-2-ARYLISOINDOLINE DIPHTHALONITRILE MONOMERS, METHODS OF MANUFACTURE, THERMOSETTING COMPOSITIONS COMPRISING THE SAME, AND USES THEREOF SHPP GLOBAL TECHNOLOGIES B.V. (NL) 2019-09-19 US disclosed
EP-3539948-A1 3-OXO-2-ARYLISOINDOLINE DIPHTHALONITRILE MONOMERS, METHODS OF MANUFACTURE, THERMOSETTING COMPOSITIONS COMPRISING THE SAME, AND USES THEREOF SABIC Global Technologies B.V. (NL) 2019-09-18 EP disclosed
EP-3539950-A1 3-OXO-2-ALKYLISOINDOLINE DIPHTHALONITRILE MONOMERS, METHODS OF MANUFACTURE, THERMOSETTING COMPOSITIONS COMPRISING THE SAME, AND USES THEREOF SABIC Global Technologies B.V. (NL) 2019-09-18 EP disclosed
EP-3539949-A1 THERMOSET 3-OXO-ISOINDOLINE DIPHTHALONITRILE POLYMERS, METHOD OF MANUFACTURE, AND USES THEREOF SABIC Global Technologies B.V. (NL) 2019-09-18 EP disclosed
US-5939508-A High temperature epoxy-phthalonitrile blends THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE NAVY (US) 1999-08-17 US disclosed
US-5389441-A Phthalonitrile prepolymer as high temperature sizing material for composite fibers THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE NAVY (US) 1995-02-14 US disclosed
US-5237045-A Heat-resistant polytriazines using acid salts of aromatic amines as catalysts for aromatic tetracyano monomers; kinetics THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE NAVY (US) 1993-08-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190284341-A1 3-OXO-2-ALKYLISOINDOLINE DIPHTHALONITRILE MONOMERS, METHODS OF MANUFACTURE, THERMOSETTING COMPOSITIONS COMPRISING THE SAME, AND USES THEREOF CYP1B1, CYP2J2, CYP1A1 LMNA 3146/4885CYP2D6 30/4885MAPK1 1326/4885
US-20190284340-A1 3-OXO-2-ARYLISOINDOLINE DIPHTHALONITRILE MONOMERS, METHODS OF MANUFACTURE, THERMOSETTING COMPOSITIONS COMPRISING THE SAME, AND USES THEREOF CYP1B1, CYP1A1, RECQL LMNA 3067/4885CYP2D6 25/4885MAPK1 1181/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.