SCHEMBL8427460

SCHEMBL8427460

CC(C=O)c1ccccc1C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACP3 P15309 1/20 0.44
HSD11B1 P28845 4/20 0.43
P2RX7 Q99572 1/20 0.43
CTSS P25774 4/20 0.40
CNR2 P34972 2/20 0.40
NFKB1 P19838 1/20 0.37
TDP1 Q9NUW8 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MC4R P32245 1/20 0.35
CTSK P43235 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27643602 0.84 CTSS (0.45) ACP3P2RX7CTSSCTSK
SCHEMBL6341623 0.82 ALDH1A1 (0.39) HSD11B1P2RX7TDP1ALDH1A1
SCHEMBL21331652 0.82 P2RX7 (0.44) ACP3HSD11B1P2RX7CNR2NFKB1
SCHEMBL29892221 0.82 ALDH1A1 (0.39) HSD11B1P2RX7TDP1ALDH1A1
SCHEMBL168980 0.81 ACP3 (0.44) ACP3HSD11B1P2RX7CTSSCNR2
SCHEMBL21495118 0.81 ACP3 (0.44) ACP3HSD11B1P2RX7CTSSCNR2
SCHEMBL14567995 0.81 P2RX7 (0.43) ACP3HSD11B1P2RX7CTSSCNR2
SCHEMBL1047625 0.78 P2RX7 (0.52) ACP3HSD11B1P2RX7CNR2TDP1
SCHEMBL84477 0.77 P2RX7 (0.50) ACP3HSD11B1P2RX7CNR2TDP1
SCHEMBL2365308 0.77 ACP3 (0.47) ACP3HSD11B1P2RX7CTSSCNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101103026-A Bicyclic heteroaryl derivatives for treating viruses GENELABS INC (US) 2008-01-09 CN disclosed
US-5973156-A Piperidine and tetrahydropyridine derivatives MERCK SHARP & DOME LTD. (GB) 1999-10-26 US disclosed
EP-0861245-A1 PIPERIDINE AND TETRAHYDROPYRIDINE DERIVATIVES MERCK SHARP & DOHME LTD. (GB) 1998-09-02 EP disclosed
WO-1997019073-A1 PIPERIDINE AND TETRAHYDROPYRIDINE DERIVATIVES MERCK SHARP & DOHME LIMITED (GB) 1997-05-29 WO disclosed