SCHEMBL8427563

SCHEMBL8427563

CCNS(=O)(=O)c1ccc(N2N=C(C)C(=CNc3ccccc3CC)C2=O)cc1.CCc1ccccc1N

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KAT8 Q9H7Z6 3/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
PTGS2 P35354 5/20 0.38
MAPT P10636 7/20 0.37
MAPK1 P28482 6/20 0.37
ALDH1A1 P00352 6/20 0.37
L3MBTL1 Q9Y468 5/20 0.37
KMT2A Q03164 5/20 0.37
MEN1 O00255 3/20 0.37
TDP1 Q9NUW8 3/20 0.37
HTT P42858 2/20 0.37
KDM4E B2RXH2 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
POLB P06746 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8427562 1.00 KAT8 (0.41) KAT8CA1CA2CA9PTGS2
SCHEMBL6950173 0.95 KAT8 (0.42) KAT8CA1CA2CA9PTGS2
SCHEMBL6950175 0.95 KAT8 (0.42) KAT8CA1CA2CA9PTGS2
SCHEMBL8015657 0.86 KAT8 (0.41) KAT8CA1CA2CA9PTGS2
SCHEMBL8015654 0.86 KAT8 (0.41) KAT8CA1CA2CA9PTGS2
SCHEMBL8428159 0.85 PTGS2 (0.46) KAT8CA1CA2CA9PTGS2
SCHEMBL8425246 0.85 L3MBTL1 (0.49) MAPTMAPK1ALDH1A1L3MBTL1KMT2A
SCHEMBL8425249 0.85 L3MBTL1 (0.49) MAPTMAPK1ALDH1A1L3MBTL1KMT2A
SCHEMBL8427580 0.84 KDM4E (0.38) KAT8CA1CA2CA9PTGS2
SCHEMBL8427578 0.84 KDM4E (0.38) KAT8CA1CA2CA9PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5869516-A 4-(arylaminomethylene)-2,4-dihydro-3-pyrazolones MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1999-02-09 US disclosed